Some Novel Benzothiazole Derivatives
Design Synthesis Characterization and Biological Evaluation of Some Novel Benzothiazole Derivatives as Anti Tubercular Agents Targeting Glutamine Synthetase 1
... OF SOME NOVEL BENZOTHIAZOLE DERIVATIVES AS ANTI-TUBERCULAR AGENTS TARGETING GLUTAMINE SYNTHETASE 1 ” submitted by the candidate bearing the Register No:261515701 in partial fulfillment of the ...
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SYNTHESIS, CHARACTERIZATION, AND ANTHELMINTIC ACTIVITY OF NOVEL BENZOTHIAZOLE DERIVATIVES CONTAINING INDOLE MOIETIES
... the benzothiazole derivatives mentioned above facts, we aimed to construct a system combining both these vital moieties such as benzothiazole and indole in a single molecular framework, together with ...
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INSILICO DESIGN, SYNTHESIS AND CHARACTERIZATION OF SOME NOVEL BENZOTHIAZOLE DERIVATIVES AS ANTI CANCER AGENTS
... Toxicity studies were carried out using ADMET SAR to determine their pharmacokinetic (ADMET) properties. A high degree of PPB implies high lipophilicity which makes the drug long-acting. All the compounds show high and ...
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Synthesis and evaluation of novel benzothiazole derivatives against human cervical cancer cell lines
... nm and at 630 nm and compared with control. The Screening for antitumor activity included measurement of results are expressed as % cell death at different conc. % cell death of EAC by tryphan blue exclusion assay. viz. ...
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Analgesic and Anti-Inflammatory Activity Studies of Some novel Benzothiazole Schiff’s bases on Experimental Rats
... of some synthesized novel benzothiazole derivatives on albino ...several benzothiazole derivatives have been ...Para-nitro benzothiazole carboxylic acid was synthesized by ...
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SYNTHESIS, CHARACTERIZATION AND BIOLOGICAL INVESTIGATION OF SOME BENZOTHIAZOLE DERIVATIVES
... A series of some novel benzothiazole derivatives were synthesized and evaluated for anti-inflammatory, antioxidant and antimicrobial activity. The structures of the compounds were confirmed by ...
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Inhibitive Effects by Some Benzothiazole Derivatives on Mild Steel Corrosion in 1 N HCl
... of some benzothiazole derivatives 1,3-benzothiazol-2- amine (BTA), 6-methyl-1,3-benzothiazol-2-amine (MBTA) and 2-amino-1,3-benzthiazole-6-thiol (TBTA) against mild steel corrosion in 1 N HCl ...
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ANTIBACTERIAL ACTIVITY OF NOVEL HYDROXY SUBSTITUTED BENZOTHIAZOLE DERIVATIVES AGAINST STREPTOCOCCUS PYOGENES
... substituted benzothiazole derivatives were first discovered in 1887 by ...reason some other methods were reported and extensively used in the laboratories that based on the use of the potassium ...
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Biological evaluation of some new 1,3-benzothiazole-2-yl derivatives containing pyrazole moiety
... Synthesis of 6-nitro-2-benzothiazolamine (2) General Procedure: A mixture of p-nitro aniline (0.01 mol) and potassium thiocyanate (0.01 mol) in 150 ml glacial acetic acid (10 %) was cooled and stirred mechanically for 30 ...
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Novel Chemical synthesis and medicinal aspects of some quinazoline and pyrimidine derivatives
... [46] Mohler, E. G.; Shacham, S.; Noiman, S.; Lezoualch, F.; Robert, S.; Gastineau, M.; Rutkowski, J.; Marantz, Y.; Dumuis, A.; Bockaert, J.; Gold, P. E.; Ragozzino, M. E. VRX- 03011, a novel 5-HT4 agonist, ...
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Synthesis of some novel thiazole derivatives
... Thiazole derivatives have attracted enormous interest due to their diverse biological ...activities. Some of them are used as ...of some substituted thiazoles are well established because of its ...
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Thiazole: A Remarkable Antimicrobial And Antioxidant Agents
... 33. Jagani CL, Sojitra NA, Vanparia SF, Patel TS, Dixit RB, Dixit BC. Microwave promoted synthesis and antimicrobial activity of 3-thiazole substituted 2-styryl- 4(3H)-quinazolinone derivatives. Journal of Saudi ...
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SYNTHESIS AND ANTIBACTERIAL EVALUATION OF BENZOTHIAZOLE DERIVATIVES
... newer derivatives of benzothiazole with enhance antibacterial ...different derivatives were synthesized. The synthesized derivatives showed very good antibacterial activities against ...
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SYNTHESIS OF SOME NOVEL THIAZOLIDINE DERIVATIVES WITH BENZOTHIAZOLE MOIETY
... As a part of systematic investigation of synthesis of N-[2-(2- chloroquinolin-3-yl)-4-oxo-1, 3-thiazolidin-3-yl]-1, 3-benzothiazole-2- carboxamide V (a-g) was achieved by corresponding manich bases IV (a-g) by ...
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SYNTHESIS AND EVALUATUION OF SOME NOVEL MERCAPTOBENZIMIDAZOLE DERIVATIVES
... has a considerable impact on antibacterial and antifungal activity. Also chloro and nitro group shows considerable effect on antiprotozoal activity. All the synthesized compounds exhibited better antiprotozoal activity ...
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A COMPREHENSIVE REVIEW ON BENZOTHIAZOLE DERIVATIVES FOR THEIR BIOLOGICAL ACTIVITIES
... Benzothiazole is a six-membered bicyclic heteroaromatic compound in which benzene ring is fused to the 4- and 5-positions of thiazole ring. Benzothiazoles are found in marine as well as terrestrial natural ...
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Cytotoxicity Analysis of Some Novel Pyrimidine Derivatives
... pyrimidine derivatives were ...that some of the compounds show moderate to good activity against bacterial and fungal stains, in which the methyl group substituted fused pyrimidine compound (4) show ...
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MULTICOMPONENT SYNTHESIS AND CHARACTERIZATION OF NEW 2 SUBSTITUTED DERIVATIVES OF 3 AMINO 4 IMINO 8 NITRO 2H PYRAZOLO [3,4 e]PYRIMIDO[2,3 b][1,3]BENZOTHIAZOLE
... substituted derivatives of 3-amino-4-imino-8-nitro-pyrazolo [3,4-e] pyrimido [2,3-b] [1,3] benzothiazole (III) obtained by the multicomponent reaction of 2-amino-6-nitro benzothiazole (I) and bis ...
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A review on Indole and Benzothiazole derivatives its importance
... Indole, Benzothiazole and its analogs research elucidated in this review furnishes the various pharmacological ...efficient derivatives with more potent therapeutic ...Indole, Benzothiazole nucleus ...
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One pot Synthesis and Antibacterial Activity of Substituted Benzothiazolyl Acetamide
... amino-6-substituted benzothiazole and pyridine was dissolved properly then added a solution of 2-hydrazino benzothiazole in pyridine and refluxed for 5 hours to give 2- [2-(1,3- benzothiazol-2-yl) ...
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