THIAZOLIDIN-4-ONE
Synthesis of 5-arylidine-2-(3, 4, 5-trimethoxyphenyl)-3-(4-phenylthiazol-2-yl) Thiazolidin-4-one Derivatives as a Novel Class of Antimicrobial Agents
... 2~(3, 4, 5~ trimethoxyphenyl)~3~(4~phenylthiazol~2~yl) thiazolidin~4~one ...of 4 with various aryl aldehydes in presence of glacial acetic acid and sodium acetate under reflux ...
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Synthesis, characterization and antimicrobial activity of some novel 2,3 disubstituted thiazolidin 4 one derivatives
... N 4 -(4-methylphenyl)-1,3-thiazole-2,4-diamine(3) was obtained by the cyclization reaction shown by the mixture of 2-chloro-N-(4-methylphenyl)acetamide and thiourea with high ...-(substituted)-N ...
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SYNTHESIS AND IN VITRO ANTIOXIDANT, ANTI INFLAMMATORY ACTIVITY OF THIAZOLYL THIAZOLIDIN 4 ONE DERIVATIVES
... 2-(2-hydroxyphenyl)-3-(4-phenyl-4,5-dihydro-1,3-thiazol-2-yl)-1,3-thiazolidin-4-one (2h) Off-white solid; M.P. 208-210ºC; Yield: 83%; λmax= 310.32; IR (KBR) cm-1: 3327 (=-C-H str.), 2928 ( ...
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Synthesis and Characterization of 2-imino-3–(2-Hydroxylphenyl)-1-Thiazolidin-4-one Substituted Ammine Complexes of Cr(III), Co(III), Ni(II) and Cu(II)
... Mixed ligand complexes of Cr(III), Co(III), Ni(II) and Cu(II) synthesized by partial substitution of 2-imino-3–(2-hydroxylphenyl)-1-thiazolidin-4-one in respective ammine complexes were characterized ...
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DESIGN, SYNTHESIS, CHARACTERIZATION OF SUBSTITUTED 3-(BENZOTHIAZOLE)-2-(PHENYL)-THIAZOLIDIN-4-ONE HETEROCYCLIC COMPOUNDS AND ITS BIOLOGICAL EVALUATION
... of thiazolidin-4- one substitute at 2 nd , 3 rd or 5 th position with active group’s posses various pharmacological activities like bactericidal ,fungicidal, hypoglycaemia, anti-malarial, ...
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ANTI BACTERIAL ACTIVITY OF 3 (4 ARYL SUBSTITUTED 3 – YL) – THIAZOLIDIN 4 – ONE AND THEIR DERIVATIVES
... RESULTS AND DISCUSSION: Based on the literature review an attempt was made to synthesize some thiazolidin-4-one compounds by microwave oven. The antibacterial screening of the synthesized compounds ...
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Synthesis, characterization and antimicrobial activity of 2,3 disubstituted thiazolidin 4 one derivatives
... three-component, one-pot synthesis of 2,3-disubstituted thiazolidin-4-one derivatives under different reaction conditions like reflux, stirring and microwave irradiation ...
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Design, synthesis and biological evaluation of novel diphenylthiazole thiazolidin 4 one based derivatives as anti inflammatory/analgesic agents
... A series of novel diphenylthiazole-thiazolidin-4-one-based derivatives was synthesized and characterized by elemental and spectral analysis. The newly synthesized compounds were screened for their ...
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ANALGESIC AND ANTI-INFLAMMATORY ACTIVITY OF NEW SUBSTITUTED THIAZOLIDIN-4-ONE DERIVATIVES Dr.Faizan Sayeed*, Abdul Sayeed, MD Akram, Mohd Waseem AkramDOWNLOAD/VIEW
... compounds. Thiazolidin-4-one has been considered as magic moiety, which is a core structure in various synthetic pharmaceuticals displaying a broad spectrum of biological ...condensed ...
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Synthesis of novel Sultams containing thiazolidin 4 one heterocycles
... 3-(2-(1,1-dioxido-1,2-thiazetidin-2-yl)ethyl)-2-(4-nitrophenyl)thiazolidin-4-one 8(f) : yield, 55%; m.p: 215-1 0 C IR (KBr) pellets reflect the molecular structure and showed the ...
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SYNTHESIS AND ANTIMICROBIAL POTENTIAL OF THIAZOLIDIN-4-ONE DERIVATIVES
... Antimicrobial evaluation by Zone of inhibition. The titled compounds thiazolidin-4-one derivatives were also screened for their antimicrobial potential against these strains by zone of inhibition. ...
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SYNTHESIS AND BIOLOGICAL ACTIVITY OF 2-(THIAZOLIDIN-4-ONE) PHENYL]-1H-PHENYLBENZIMIDAZOLES AND 2-[4-(AZETIDIN-2-ONE)-3-CHLORO-4- PHENYL] -1H-PHENYL BENZIMIDAZOLES
... A new series of 2-[4-(azetidin-2-one)-3-Chloro-4-phenyl]-1H-Phenylbenzimidazoles and 2-(thiazolidin-4-one)-Phenyl]- 1H-Phenylbenzimidazoles were synthesized by the reaction of ...
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MICROWAVE ASSISTED SYNTHESIS OF SOME NEW THIAZOLIDIN 4 ONE DERIVATIVES CONTAINING A PYRIMIDONE AND QUINOLINE MOITIES
... on thiazolidin-4- one derivatives I am reporting the synthesis 6-Methyl-2-oxo/thioxo-4-(substituted) phenyl-1, 2, 3, 4-tetrahydro-pyrimidine-5-carboxylic acid ...
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DESIGN, SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF NEW SUBSTITUTED THIAZOLIDIN-4-ONE DERIVATIVESDr. Faizan Sayeed*, Abdul Sayeed, MD Akram, Mohd Waseem AkramDOWNLOAD/VIEW
... compounds. Thiazolidin-4-one has been considered as magic moiety, which is a core structure in various synthetic pharmaceuticals displaying a broad spectrum of biological ...condensed ...
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THIAZOLIDIN-4-ONE DERIVATIVES ON HUMAN LUNG FIBROBLAST SHOWS OXYGEN FREE RADICAL SCAVENGING ACTIVITY
... The antioxidants are proving crucial tools in the exploration of oxidant stress-related diabetic pathologies and despite the noticeable prospective merit of the safety and efficacy of antioxidant supplementation in any ...
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Hyperglycedemia and hypertriglyceridemia activities of newly synthesized compounds derived from 3'-(4-halophenyl)-5'-arylidene spiro(cyclohexane- (1,2')-thiazolidin)-4'-one
... 5-Arylidene spiro[cyclohexane-(1,2')-thiazolidin-4'-one derivatives 1a-d were treated with some nucleophiles. So, when 1b was treated with hydrazine hydrate or phenylhydrazine it gave the ...
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Synthesis Characterization and Pharmacological Activity of Novel Thiazolidin – 4 one Analogues
... synthesized compounds was carried out by MES induced convulsions method using albino mices of either (20-30 g). animals were deprived of food for 18hrs. prior to experiment (the first group was control group and received ...
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Synthesis, Characterization and Study of Liquid Crystalline Behavior of New Compounds Containing Thiazolidin-4-one, 1, 2, 3-Triazole and Benzimidazol Rings
... Synthesis of 1,1-((1,3 Phenylenebis (Azanediyl)) Bis (2-Oxoethane-2,1- diyl))Bis(4,5-Dihydro-1H-1,2,3-Triazole-4- Carbonyl Chloride) [VI] and 1,1- ((1,3 Phenylenebis (Azanediyl)) Bis (2- Oxoethane-2,1-diyl)) Bis ...
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Journal of Applied Pharmaceutical Science
... IR spectra of compounds 9a,b revealed characteristic bands at 1732, 1697 cm -1 , respectively, which correspond to the carbonyl group of the 1,3-thiazolidin-4-one ring. 1 H-NMR spectra of compounds ...
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Synthesis and Characterization of the Thiazolidinone and/or Thiourea substituted Amine Complexes of Cu (II)
... Mixed ligand complexes of copper (II), involving either Mercaptyl thiazolidinone (1) [2-(2- hydroxy benzoyl)-3-N-(2-mercaptyl)-1-Thiazolidin-4-one] or Pyridine thiazolidinone (2) [ 2-(2- hydroxy ...
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