[PDF] Top 20 BENZOTHIAZOLE DERIVATIVE: A REVIEW ON ITS PHARMACOLOGICAL IMPORTANCE TOWARDS SYNTHESIS OF LEAD

... In 2016 Rosales-Hernandez MC et al, synthesized some benzothiazole derivatives Fig. 30 and evaluated their antioxidant activity. In their study, they found that compound (E)-5-((benzo[d]thiazol- 2-ylimino) (methyl ... See full document

... diverse pharmacological and biological ...acid. Benzothiazole is one of the most important heterocyclic compound, weak base, having varied biological activities and still of great scientific interest now a ... See full document

... finds its use as one of the major parts in pharmaceutical chemistry as useful biological entities and improved pharmacological ...diversified pharmacological activities and their analogues are known ... See full document

... The oxadiazole dr ugs were the first effective chemotherapeutic agents to be employed systematically for the prevention and cure of bacterial infection in human beings. Benzothiazole with oxadiazole groups were ... See full document

... in Pharmacological activities: Imidazole derivatives have a wide range of pharmacological ...and its derivative are reported to have, analgesic and anti-inflammatory activity, cardiovascular ... See full document

... A series of new benzothiazole derivatives have been synthesized, in five steps, from substituted phenols via the 1,3,4-oxadiazole-2-thiones .The in vitro antitumor activity of the compounds obtained was ... See full document

... 13. Anti-Ulcer: Acute gastric ulcers were induced in rat model by cold restraint stress, pyloric ligation, aspirin plus pyloric ligation, and duodenal ulcers induced by cysteamine. The protective activity of the extract ... See full document

... 10 min were recorded by placing the animals in the actophotometer, which gives the initial reading. The compounds were administered intraperitonially in the form of suspension prepared in 1% Tween-80 at a dose of 30 ... See full document

... Some 1-{4-Chloro-6-[3-(6-methoxy - benzothiazol-2-ylazo)-2,6-dimethyl-quinolin-4-yloxy]- [1,3,5] triazin-2-yl}-(substituted phenyl)-urea 3a-h were synthesized and studied for their microbial activity. These compounds ... See full document

... for its medicinal properties since the Bronze age (3000 - 2000 ...various pharmacological activities as antioxidants, analgesic, anti-inflammatory, anti-ulcer, anti-viral, immuno-modulatory, ... See full document

... Ailantinol E, ailantinol F, and ailantinol G, and related compounds isolated from Ailanthus altissima grown in Taiwan, were evaluated for its antitumor promoting effects against Epstein-Barr virus early antigen ... See full document

... oxadiazole derivative of 28-carbomethoxy lupan [2,3-C]-1’, 2’, 5’-oxadiazole 6 with respect to parent compound Betulinic acid 1 tested in disc diffusion ...oxadiazole derivative 6 maximum inhibition was ... See full document

... Various substituted 3-{7-substituted-6-1,3 -benzothiazol-2-yl-1-({4-methylphenyl) sulfonyl]20thixo-2,3dihydroquinazolin –4 (1H)-one and 2-[(4Z)-4-benzylidine-2-phenyl-5-oxo-4,5- ... See full document

... pot synthesis of 3-amino-4-imino-8-methoxy- (2H) Pyrazolo [3’,4’;4,5] pyrimido[2,1-b] benzothiazole and its 2-substituted derivatives is convenient over tradinational rout of synthesis of this ... See full document

... complexes of heterocyclic compounds and their Ni (II), Pd (II), Pt (I), Cu (II) complexes have also been synthesized. Heterocyclic r ing system like benzothiazole and few metals like Zn (II,) Pt (II), Cu (II), Ni ... See full document

... Manin-Darby canine kidney (MDCK) cells were trans- fected with cDNA APP with a 42 amino acid truncation at the C-terminus (DeltaC). A unique Aβ sequence was found and immunoprecipitated with an Aβ 17-24-specific ... See full document

... This study indicates that the production of DHAQC (2) warranted a better yield (32%) than the synthesis of damnacanthal. The synthesized DHAQC (2) also possessed better selectivity against estrogen-dependent ... See full document

... People are settling for remedies that are not just effective but are harmless in the long run. Herbal oils are of various types depending on herbs used to extract the oil. The most important bioactive constituents of ... See full document

... have its origin in the Greek (agremone), which refers to plants which supposedly healed cataracts of the ...remedies. Its ancient uses include treatment for catarrh (mucous membrane inflammation with ... See full document

... 2015 Various Plant Parts of Anacardium occidentale L was carried out to evaluate the presence of anacardic acid, total phenolic compound, antioxidant activity and antibacterial activity in methanolic extract of callus ... See full document