[PDF] Top 20 Discovery and evaluation of novel anti-inflammatory derivatives of natural bioactive curcumin
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Discovery and evaluation of novel anti-inflammatory derivatives of natural bioactive curcumin
... of curcumin and estimated their anti- inflammatory activities against LPS-induced TNF- α and IL-6 release in mouse ...monocarbonyl curcumin analogs with symmetric and heterocyclic structures ... See full document
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Studies of synthetic chalcone derivatives as potential inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and pro-inflammatory cytokines
... chalcone derivatives, 1b was the strongest inhibitor of sPLA 2 -V with IC 50 ...Major anti-inflammatory agents, steroids, and COX, were proven to have serious side effects so now attention is toward ... See full document
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Synthesis and evaluation of novel pyrrolidine chalcone derivatives with anticancer, anti inflammatory and antibacterial activities
... Serious infections caused by microorganisms resistant to commonly used antimicrobials have become a major healthcare problem worldwide in the 21 st century. This is responsible for the significant increase in morbidity ... See full document
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Synthesis and Evaluation of Novel 1, 5-Benzothiazepine Derivatives as Anti-Inflammatory Agents
... various bioactive heterocycles and green methods, which is applicable in organic ...of bioactive heterocyclic compound and designation of green chemical reactions and their applications in organic ... See full document
8
SYNTHESIS AND BIOLOGICAL EVALUATION OF SOME NOVEL CHALCONE DERIVATIVES AS ANTI INFLAMMATORY AGENTS
... of natural products and are considered as the precursors of flavonoids and ...its derivatives represent one of the most active classes of heterocyclic compounds possessing a wide spectrum of biological ... See full document
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Design, Synthesis, and Anti-Inflammatory Activity of Novel Quinazolines
... synthetic derivatives, but also in several naturally occurring alkaloids isolated from animals, plants, and microorganisms, for example, tryptahthin and ...non-acidic anti-inflammatory drugs 1,2 ... See full document
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ANALGESIC AND ANTI INFLAMMATORY ACTIVITIES OF NOVEL THIAZINE DERIVATIVES
... analgesic, anti anxiety, anti-inflammatory ...thiazine derivatives have been the subject of chemical and biological studies on account of their interesting pharmacological ...Such ... See full document
10
Anti-inflammatory Activities of Novel Derivatives of Hydrazide- Hydrazones
... hydrazones derivatives were characterized by CHN analyses, IR, and 1 H NMR spectral ...their anti-inflammatory activity. All compound exhibited anti-inflammatory activity at the dose ... See full document
5
Synthesis and antimicrobial evaluation of novel 1,2,4-triazine derivatives
... 5-(4-fluorobenzyl)-3-(furan-2-yl)-1,2,4-triazin-6(1H)-one 4 was synthesized. Treatment of the latter with POCl 3 afforded the chloro derivative 5. Hydrazinolysis of compound 5 with hydrazine hydrate in ethanol yielded ... See full document
6
Synthesis and Screening of Anti-inflammatory Activity of Benzofuran Derivatives Bearing Oxadiazole
... In conclusion, several benzofuran analogs of fenamates were synthesized. These compounds contain benzofuran moiety instead of benzene moiety which is present in fenamates. Further the carboxylic acid moiety was conver ... See full document
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SYNTHESIS, CHARACTERIZATION, ANTIOXIDANT AND ANTI-INFLAMMATORY ACTIVITY EVALUATION OF SOME SUBSTITUTED PYRAZOLE DERIVATIVES
... ABSTRACT: A series of substituted acetophenones are condensed with hydrazides to the corresponding hydrazones which are subsequently cyclized by using volumizer-Haack reaction to give new pyrazole derivatives. All ... See full document
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Anti-Inflammatory Activity Of Novel 1,2-Dihydroquinoline Derivatives
... Sub-planter injection of carrageenan to left hind paw of rats resulted in significant (p<0.01; p<0.001) increase in paw volume at different tested time intervals compared to normal control animals. Administration ... See full document
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ANTI-INFLAMMATORY EVALUATION OF SOME NOVEL SUBSTITUTED- [1,2,4] TRIAZOLO[1,5C]QUINAZOLINONE DERIVATIVES
... search novel anti-inflammatory heterocyclic in the condensed quinazolinone series, representative compounds were synthesized via a suitable reaction ... See full document
7
Synthesis of some benzoxazole derivatives and their anti inflammatory evaluation
... benzoxazole derivatives throughthe reaction of substituted 2-aminophenols and acyl chlorides in the presence ofcatalytic amount of In(OTf)3 under solvent-free reaction ... See full document
8
Synthesis and Biological Evaluation of Quinazolinone Fused Chalcone Derivatives as Anti-inflammatory Agents
... PC, Roth BD, Beylin VG, Gilbertsen RB, Chan K, Schrier DJ, Guglietta A, Bornemeier DA, Dyez RD. Synthesis, structure-activity relationships, and in-vivo evaluations of substituted di-tert- butylphenols as a novel ... See full document
6
Synthesis and Antibacterial Evaluation of Some Novel Chalcones and their Derivatives
... In view of the above and in continuation of our work 10-12 on chalcones and its derivatives, we herein report a new series of chalcones (6a-e), acetylpyrazolines (7a-e) aminopyrimidines[r] ... See full document
5
Evaluation of Anti-Propionibacterium Acnes and Anti-Inflammatory Effects of Polyphenolic Extracts of Medicinal Herbs in Jordan
... the anti-inflammatory effects of the selected herbs, Arum exhibited a unique potent inhibitory effects on the release of IL-1a pro-inflammatory ...the anti-inflammatory effect of Arum ... See full document
7
Synthesis and anti inflammatory study of novel fluorobenzothiazole derivatives
... Benzothiazole belongs to an important class of heterocyclic compounds and exhibits a wide range of biological properties and due to its potent activities, thus the synthesis of benzothiazole is an area of current ... See full document
15
Synthesis of 2-Substituted-4,6-Diphenylpyridazinones as Potent Anti-Inflammatory Agents
... Rats were killed under deep ether anesthesia 24h after the anti-inflammatory experiment, and their stomachs were removed. The abdomen of each rat was opened through great curvature and examined for lesions ... See full document
10
Discovery and evaluation of asymmetrical monocarbonyl analogs of curcumin as anti-inflammatory agents
... ger anti-inflammatory activity compared with the leading compound ...the anti-inflammatory activity of the most active compounds, 3a and ...monocarbonyl curcumin analogs may be utilized ... See full document
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