[PDF] Top 20 SYNTHESIS AND BIOLOGICAL EVALUATION OF SOME NOVEL CHALCONE DERIVATIVES AS ANTI INFLAMMATORY AGENTS
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SYNTHESIS AND BIOLOGICAL EVALUATION OF SOME NOVEL CHALCONE DERIVATIVES AS ANTI INFLAMMATORY AGENTS
... All reagents and solvents for synthesis were obtained from Alfa Aesar and Sigma-Aldrich chemicals. All materials used for this experiment are analytical grade. Melting points of the products were determined in ... See full document
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Synthesis and Biological Evaluation of Andrographolide Derivatives as Potential Anti-Inflammatory Agents
... Zhang Z, Wang Y, Xu L, Yu P. Synthesis and biological evaluation of andrographolide derivatives as potential anti- inflammatory agents. J Pharm Biomed Sci ... See full document
6
SYNTHESIS AND BIOLOGICAL EVALUATION OF COUMARIN DERIVATIVES AS ANTI INFLAMMATORY AGENTS
... Synthesis of 7-hydroxy- 4-methyl coumarin: A beaker containing 100 ml of concentrated sulphuric acid was kept in an ice bath, to this solution 0.1 mol of resorcinol and ethyl acetoacetate was added, with ... See full document
8
Synthesis, characterization and biological evaluation of novel 1,2,4-triazole derivatives as potent antibacterial and anti-inflammatory agents
... The synthesized compounds Carrgennan-induced mice paw oedema test for acute inflammation, the synthesized compounds 3-(biphenyl-4-yl)-4-(2-chloro-5-(trifluoro methyl) phenyl)-1H-1,2,4-triazole-5(4H)-thione (R12), 3- ... See full document
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Synthesis and biological evaluation of some new coumarin derivatives as potential antimicrobial, analgesic and anti inflammatory agents
... Melting points were determined on an electro thermal melting point apparatus [Stuart Scientific, model SMP3, England, UK], and were uncorrected. A pre-coated silica gel plate (kieselgel 0.25 mm, 60G F254, Merck, Germany) ... See full document
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Synthesis and biological evaluation of a novel class of curcumin analogs as anti-inflammatory agents for prevention and treatment of sepsis in mouse model
... The anti-inflammatory activity of compound 3f is likely via downregulating NF- κ B and ERK pathways, and blocking I κ B ...exert anti-inflammatory activities by different mechanisms, which are ... See full document
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Synthesis and Biological Evaluation of Some Piperazine Derivatives as Anti-Inflammatory Agents
... for anti- inflammatory activity by inhibition of carrageenan induced rat paw edema method at the dose of 10 ...Significant anti-inflammatory activity was observed with inhibition in the range ... See full document
6
Synthesis, Biological Evaluation and Molecular Modeling Studies of Some 5 Methylisoxazole Derivatives as Anti Inflammatory Agents
... Some novel 4-(5-methylisoxazol-3-ylamino) thiazole derivatives incorporated with different heterocyclic moieties were synthesized and screened for their anti-inflammatory ...their ... See full document
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Synthesis and Biological Evaluation of Quinazolinone Fused Chalcone Derivatives as Anti-inflammatory Agents
... RD. Synthesis, structure-activity relationships, and in-vivo evaluations of substituted di-tert- butylphenols as a novel class of potent, selective, and orally active cyclooxygenase-2 inhibitors: ... See full document
6
Synthesis and evaluation of novel pyrrolidine chalcone derivatives with anticancer, anti inflammatory and antibacterial activities
... the synthesis of compounds(3AP-3JP) is mentioned in the scheme ...pyrrolidin-1-yldiazenyl]phenyl}ethanone synthesis was done by following the common procedure for the coupling reactions of diazonium ... See full document
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SYNTHESIS, CHARACTERIZATION AND BIOLOGICAL EVALUATION OF SOME NEW HETEROCYCLIC DERIVATIVES OF CHALCONE AS ANTIHYPERGLYCEMIC AGENTS
... . Anti-Hyperglycemic Activity (Effect on Sucrose Loaded Diabetic Model): All the compounds were evaluated for their in-vivo ant hyperglycemic activity using sucrose loaded diabetic model and fall in blood glucose ... See full document
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SYNTHESIS AND BIOLOGICAL EVALUATION OF CHALCONE DERIVATIVES OF ACRIDINES AS ANTICANCER AGENTS
... synthetic chalcone fused acridine derivatives (10a-j) was evaluated on three human cancer cell lines such as MCF-7 (Beast), A549, MDA MB-231 (lung) by using the MTT assay and these results are summarized in ... See full document
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EVALUATION OF ANTI-INFLAMMATORY ACTIVITIES OF NEWLY SYNTHESIZED ISATIN DERIVATIVES IN RATS
... On the other hand, Carbamate-bearing molecules has found to have an interesting role in modern drug discovery and medicinal chemistry. Organic carbamates (or urethanes) are structural elements of many approved ... See full document
6
Design Synthesis Characterization and Biological Evaluation of Some Novel Benzothiazole Derivatives as Anti Tubercular Agents Targeting Glutamine Synthetase 1
... In any docking scheme, two conflicting requirements must be balanced: the desire for a robust and accurate procedure, and the desire to keep the computational demands at a reasonable level. The ideal procedure would find ... See full document
118
Synthesis and biological evaluation of some novel isatin derivatives as antimicrobial agents
... spirooxindole derivatives were synthesized by the one-pot three component reaction involving isatin, malononitrile and cyclic 1,3-diketo compound using TBAB as a novel and inexpensive catalyst in ethanol ... See full document
5
Synthesis and Biological Evaluation of Substituted Pyrazoline Derivatives Bearing 3,4,5 Trimethoxyphenyl Moiety as Anticancer, Anti inflammatory and Antioxidant Agents
... Inflammation is body’s way of dealing with infection and tissue damage, but there is a fine balance between the beneficial effects of inflammation cascades and their potential for long-term tissue destruction. If they ... See full document
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SYNTHESIS AND BIOLOGICAL EVALUATION OF SOME NOVEL HETEROCYCLIC CHALCONE DERIVATIVES
... In the present work chalcones were used to prepare various heterocyclic compounds by cyclization with urea/thiourea/2,4-dinitrophenylhydrazine in presence of ethanolic sodium hydroxide/ sodium acetate gives good yields. ... See full document
5
INSILICO DESIGN AND MOLECULAR DOCKING STUDIES OF NOVEL 1, 2, 4- TRIAZOLE DERIVATIVES AS CYP-51 INHIBITORS
... triazole derivatives have been studied extensively owing to their interesting biological activities such as antibacterial [1,2] , antifungal [3] , antiviral [4,5] , anti convulsant [6] , anti- ... See full document
9
Design, Synthesis, Characterization and Biological Evaluation of Some Novel Butyrolactone Derivatives of Chalcone as Antitubercular Agents.
... the biological target obtained through methods such as x-ray crystallography or NMR ...the biological target, candidate drugs that are predicted to bind with high affinity and selectivity to the target may ... See full document
85
Studies of synthetic chalcone derivatives as potential inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and pro-inflammatory cytokines
... the chalcone derivatives, 1b was the strongest inhibitor of sPLA 2 -V with IC 50 ...Major anti-inflammatory agents, steroids, and COX, were proven to have serious side effects so now ... See full document
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