2-(4'-AMINOPHENYL)BENZOTHIAZOLE
Synthesis, Biological Evaluation of 4 aminoquinoline 1, 2, 4 triazole Conjugated Benzothiazole as Potent Analgesic, Anti inflammatory
... of 4-aminoquinoline so we had designed and synthesized the 4-(Substituted Benzothiazol-2-ylamino)-5-[2-(7-chloro- quinolin-4-yl amino)-ethyl amino] substituted ...
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SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF 2 SUBSTITUTED BENZOTHIAZOLE DITHIOMIDOCARBONATE DERIVATIVES
... 2-amino benzothiazole (0.025 mole) and aqueous sodium hydroxide solution (10M, 4ml) were stirred in 10 ml of dimethyl formamide for 15 minutes then carbon disulpide was added drop wise the reaction mixture ...
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Multicomponent Synthesis and Pharmacological Screening of 3-Cyano -4-Imino -2- Methylthio -8- Nitro -4H- Pyrimido [2,1-b] [1,3] Benzothiazole and its 2-Substituted Derivatives
... [2,1-b] benzothiazole and its 8- substitued derivatives were synthesized by Nair Mohan ...[2,1-b] benzothiazole) carboxylic acids and esters has been reported by Alaimo Robert ...containing ...
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MULTICOMPONENT SYNTHESIS AND CHARACTERIZATION OF NEW 2 SUBSTITUTED DERIVATIVES OF 3 AMINO 4 IMINO 8 NITRO 2H PYRAZOLO [3,4 e]PYRIMIDO[2,3 b][1,3]BENZOTHIAZOLE
... 1) Synthesis of 3-amino-4-imino-8-nitro-2H-pyrazolo[3,4-e]pyrimido[2,3-b][1,3] benzothiazole (a): A mixture of 2-Amino-6-nitro benzothiazole [0.195 gm, 0.001 mole], bis methylthio methylene ...
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Synthesis, characterization and biological activities of 2 aryl 3 substituted 4 thiazolidinones carrying benzothiazole moiety
... During recent years there has been considerable interest in the development of novel compounds with anticonvulsant, antidepressant, analgesic, anti-inflammatory, antiallergic, antipsychotic, antimicrobial, ...
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Crystal Structure of 2 [2 (4 Methylphenyl)Ethenyl] 1,3 Benzothiazole
... atoms. Benzothiazole is an important scaffold with a wide array of interesting biological activities and therapeutic ...applications. Benzothiazole derivatives have emerged as significant components in ...
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Synthesis and pharmacological evaluation of azetidin-2-ones and thiazolidin-4-ones encompassing benzothiazole
... Various 7-chloro-6-fl uoro-2-arylidenylaminobenzo(1,3)thiazole (2a-h) have been synthesized by the condensation of 7-chloro-6-fl uoro-2-aminobenzo(1,3)thiazole (1) with different aromatic aldehydes. The ...
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Synthesis and Characterization of Palladium(II) Complexes with 2-(2′-hydroxylphenyl)benzoxazole, 2-(2′-hydroxyl phenyl)benzothiazole or the Mixed Ligands
... [PdCl 2 (Hpbo) 2 ], trans-[PdCl 2 (Hpbt) 2 ] or trans-[PdCl 2 (Hpbo)(Hpbt)], respectively the benzoxazole or benzothiazole ligands behave as monodentate ligands coordinated to ...
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SYNTHESIS OF SOME NOVEL THIAZOLIDINE DERIVATIVES WITH BENZOTHIAZOLE MOIETY
... ethyl- 2-benzthiozole ...3- benzothiazole-2-carbohydrazide. 2-methylquinoline-3-carbaldehyde reflux with 1,3- benzothiazole-2-carbohydrazide gives ...
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Biological important Co(II) ternary complexes of 2 substituted benzazoles and amino acids
... and benzothiazole have gained importance because of their biological significance ...and benzothiazole and their derivatives have been reported by Seth et ...
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A convenient one pot synthesis of some novel benzothiazole and its derivatives
... pyrimido[2,1-b] benzothiazole and its 2-substituted derivatives is convenient over tradinational rout of synthesis of this organic ...3-cyno-4-imino- 2-methylthio-8-methoxy-4H-pyrimido [2,1-b] ...
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Benzothiazole: Unique and versatile scaffold in the field of cancer
... novel benzothiazole-2-thiol derivatives, and they were evaluated for anticancer ...linked benzothiazole-2-thiol compounds 7d, 7e, 7f and 7i exhibited potent and broad-spectrum inhibitory ...
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Analgesic and Anti-Inflammatory Activity Studies of Some novel Benzothiazole Schiff’s bases on Experimental Rats
... 6-carboxy-2-(P-aminophenyl) benzothiazole: 6-carboxy-2-(P-nitrophenyl) benzothiazole ...MgSO 4 , filtered and concentrated to a solid that was triturated ...
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Synthesis of Fluoro Substituted Benzothiazoles Incorporated with 1,3,4-Thiadiazoles for Biological and Pharmacological Screening
... substituted 2[5'-(3-Methyl benzene)-1',3',4-thiadiazol-2'-yl amino)-6-flouro-7substituted (1,3) benzothiazoles and 2[5'-(p-chlorobenzene)-1',3',4'-thiadiazole-2'-yl amino) ...
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Synthesis, biological and pharmacological activities of 2 methyl 4H pyrimido[2,1 b][1,3]benzothiazoles
... substituted 2-amino[2,1-b][1,3]benzothiazoles ...yielded, 2-methyl-4-H-pyrimido[2,1- b][1,3]benzothiazole-4-ones 4a-h and ethyl 4-phenyl-2-methyl-4H–pyrimido[2,1- ...
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BENZOTHIAZOLE ITS CURRENT PHARMACOLOGICAL PROFILE AND METHODS OF SYNTHESIS
... substituted 2-(4- aminophenyl) benzothiazoles, were developed and comprised a novel class of antitumor active compounds, especially against sensitive breast tumor cell lines, ...new 2-Amino ...
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Synthesis and characterization of transition metal complexes with newly synthesized substituted benzothiazole
... compound, 4-bromo-2-hydrazino-6-methyl benzothiazole and different experiments were conducted to see the chelating tendency of newly synthesized heterocyclic ...When ...
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ANTIFUNGAL ACTIVITY OF PYRIMIDO BENZOTHIAZOLE DERIVATIVES BY DISC DIFFUSION METHOD
... [1,3] benzothiazole and its 2-substituted derivatives are responsible for antifungal activity, but it is interesting to note that benzothiazole moieties when fused with other moieties showed a broad ...
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A FACILE SYNTHESIS AND BIOLOGICAL EVALUATION OF SOME MACROCYCLIC COPPER COMPLEXES
... of 2-amino 6- bromo benzothiazole: 2-amino 6-bromo benzothiazole was synthesized using thiocyanogenation ...(Na 2 CO 3 ) is added to neutralize it, till the solid was ...
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“Synthesis of Oxadiazole Derivatives: An Overview” by Leena K Pappachen, Amrutha Unnikrishnan, Revathy Sreedhar, Shalumol A, Sneha James, India.
... To a solution of anthranilic acid (0.05mole, 6.85g) in ethanol, conc. sulphuric acid was added dropwise and shaked for few min till a white coloured precipitate of ethyl-2-aminobenzoate was formed. To this, ...
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