adrenergic receptor
Effects of three beta adrenergic receptor agonists on growth performance, blood biochemical parameters, fatty acids composition and carnitine palmitoyltransferase I gene expression of rainbow trout, Oncorhynchus mykiss
... beta adrenergic receptor agonists studies on growth performance of fish species; except two reports (Lortie et ...beta adrenergic agonists. For example, salbutamol (a beta 2 adrenergic ...
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Topical administration of adrenergic receptor pharmaceutics and nerve growth factor
... -adrenergic receptor antagonists produce retinal dysfunction, we have also recently found that β -adrenergic receptor agonists are beneficial to the ...
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The Roles of β-Adrenergic Receptor Blockers in Interstitial Cystitis
... β-Adrenergic receptor blockers appear to have a beneficial clinical effect in ...β- adrenergic receptor blockade and ...β- adrenergic receptor blockade to IC ...
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Adrenergic receptor control mechanism for growth hormone secretion
... Alpha adrenergic blockade with phentolamine during insulin hypoglycemia, ...Beta adrenergic blockade with propranolol during insulin hypoglycemia significantly enhanced HGH concentrations in paired ...alpha ...
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The Role of Beta-Adrenergic Receptor Blockers in Autism
... β-adrenergic receptor is conferred may increase the risk for alterations, such as those that that lead to autism, in ...β-adrenergic receptor polymorphisms in individuals with ...
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Biphasic Adrenergic Modulation of β Adrenergic Receptors in Man: AGONIST INDUCED EARLY INCREMENT AND LATE DECREMENT IN β ADRENERGIC RECEPTOR NUMBER
... that adrenergic agonists modulate the number of available b-adrenergic receptors on circulating mononuclear cells in a biphasic manner, with an early increment and a late decrement, in ...
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Myocardial beta adrenergic receptor function during the development of pacing induced heart failure
... beta-adrenergic receptor density was not changed at any time point, but beta 1-adrenergic receptor density was decreased (P < ...beta-adrenergic receptor dysfunction in ...
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Rapid desensitization of neonatal rat liver beta adrenergic receptors A role for beta adrenergic receptor kinase
... of receptor responsiveness. The proposed mechanisms of such rapid receptor desensitization include receptor phosphorylation by either cAMP-dependent protein kinase or the specific ...
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Anti–β1 adrenergic receptor antibodies and heart failure: causation, not just correlation
... Antibodies specific for the b 1 -adrenergic receptor are found in patients with chronic heart failure of various etiologies. From work presented in this issue of the JCI, we can now infer that these ...
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Effects of Adrenergic Receptor Activation and Blockade on the Systolic Preejection Period, Heart Rate, and Arterial Pressure in Man
... ventricle. The preejection period was determined from high speed, simultaneous recordings of the phonocardiogram, carotid pulse tracing, and electrocardiogram. The preejection period was shortened by isoproterenol, ...
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Original Article Relationship between the β1-adrenergic receptor and the β2-adrenergic receptor in hypertension
... Abstract: Objective: To determine whether β1 adrenergic receptor (β1-AR) changes are related to β2-AR expression under conditions of hypertension. Methods: The mRNA and protein levels of β1- and β2-AR in ...
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Beta adrenergic receptor polymorphisms: A basis for pharmacogenetics
... Medical therapy with β-blockers has been used for more than a half a century for the treatment of most car- diovascular diseases, such as acute myocardial infarction, chronic coronary artery disease, arterial ...
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Interaction between Antagonist of Cannabinoid Receptor and Antagonist of Adrenergic Receptor on Anxiety in Male Rat
... α2 adrenergic receptor antagonist) caused a decrease in CB1 receptor density in the PFC, suggesting that high extracellular level of nor- epinephrine down regulates CB1 receptors (Hardy, ...CB1 ...
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Reduced beta adrenergic receptor activation decreases G protein expression and beta adrenergic receptor kinase activity in porcine heart
... beta-adrenergic receptor-G-protein-adenylyl cyclase pathway in porcine ...cardiac adrenergic signaling associated with chronic reduction in beta- adrenergic receptor agonist activation ...
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An antiidiotypic antibody that recognizes the beta adrenergic receptor
... adrenergic receptor. Allotype-identicaL rabbits were immunized with this fraction. After 6 mo, antisera exhibited antiidiotypic activity inhibiting [3H]alprenolol binding to the original antibody and to ...
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Inhibition of p38α MAPK rescues cardiomyopathy induced by overexpressed β2 adrenergic receptor, but not β1 adrenergic receptor
... We examined the role of p38a MAPK in mediating cardiomyopathy in mice overexpressing b 1 -adrenergic receptor (b 1 -AR) or b 2 -AR by mating them with dominant-negative p38a (DNp38a) MAPK mice. Both b 1 -AR ...
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Polymorphisms of the 5' leader cistron of the human beta2 adrenergic receptor regulate receptor expression
... pranolol in the aforementioned buffer for 2 h at 25 8 C. The reaction was stopped by dilution and rapid vacuum filtration over Watman GF/C filters. Radioactivity was measured in a gamma counter at 80% efficiency. Protein ...
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The Glucose Receptor A DEFECTIVE MECHANISM IN DIABETES MELLITUS DISTINCT FROM THE BETA ADRENERGIC RECEPTOR
... beta adrenergic receptors and the implications of this relationship with regards to abnormal insulin secretion in diabetes mellitus, two questions were ...beta adrenergic activity, the effect of beta ...
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Molecular characterization of [beta]2 adrenergic receptor haplotypes
... 16 receptor undergoes enhanced agonist-promoted down-regulation in receptor number in comparison to the Arg 16 ...27 receptor undergoes very little agonist-promoted down-regulation compared to the ...
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A New and Alternate Synthesis of Carvedilol: An Adrenergic receptor
... A New and alternate synthesis of carvedilol, β-adrenergic blocking agent is reported and finalized the meritorious one. The key step in this approach is synthesis of o-protected 1-(9H- ...
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