Antitubercular Activity
Synthesis and antitubercular activity of some new 2, 3 disubstituted quinazolinones
... of activity and drug resistant pathogens, especially Mycobacterium tuberculosis a series of 2-(substituted)-N-(4oxo-2-(pyridine-2- yl)quinazolin-3(4H)-yl acetamide and 2 ...
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Synthesis and evaluation of antitubercular activity of some thiobenzimidazolyl derivatives
... spectra. Antitubercular activity was evaluated for synthesized compounds; most of them reported good antitubercular activity against Mycobacterium ...
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SCREENING OF ABUTILON INDICUM L LEAF AND SEED EXTRACTS FOR ANTITUBERCULAR ACTIVITY
... the Antitubercular activity of Abutilon indicum ...invitro Antitubercular activity using Microplate Alamar Blue Assay against Mycobacterium tuberculosis H37Ra and Mycobacterium bovis ...
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DESIGN, SYNTHESIS AND EVALUATION OF ANTITUBERCULAR ACTIVITY OF AMINO AZETIDINONES FROM ISONIAZID
... known antitubercular drug isoniazid not only as a mode to improve its antitubercular activity but also to minimize other problems associated with INH ...study antitubercular effect, the one ...
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Solution Phase Synthesis of Small Schiff Bases Combinatorial Library with Potential Antitubercular Activity
... their antitubercular activity against four Mycobacterium ...anti-TB activity was revealed with the investigated mixtures and maximum activity shown by M 2 and M 7 at a concentration of ...
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In vitro screening of quinoxaline 2 one derivatives for antitubercular activity
... A series of ethyl 2-[(3-methyl-2-oxoquinoxalin-1(2H)-yl)acetyl]-3-oxo-2,3-dihydro-1H- pyrazole-4-carboxylate derivatives were prepared and evaluated for their antitubercular activities. All compounds were screened ...
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Synthesis and antitubercular activity of some novel N-methyl triazolone derivatives
... for antitubercular activity. In the antitubercular activity studies, of these compounds P4 and P5 showed very significant activity and P1, P2, P3 showed moderate antitubercular ...
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ANTI MRSA AND ANTITUBERCULAR ACTIVITY OF PHENOXAZINONE CONTAINING MOLECULE FROM BORRA CAVES STREPTOMYCES SP BCA1
... It is known that actinobacteria are dominant among the heterotrophic bacterial population present in caves 8 . However, only limited works are carried out on actinobacteria from Indian caves in terms of biodiversity and ...
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Synthesis, antitubercular activity and mechanism of resistance of highly effective thiacetazone analogues
... Our previous work demonstrated that in M. bovis BCG, M. chelonae and M. marinum, TAC inhibits the methyltransferases that introduce cyclopropane rings into mycolates [20]. Members of this methyltransferase family of ...
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PHYTOCHEMICAL ANALYSIS AND ANTITUBERCULAR ACTIVITY OF FLOWERS EXTRACT OF MANGIFERA INDICA
... ABSTRACT: About 5 extract (hexane, acetone, ethanol, methanol, aqueous extraction) from the flowers of Mangifera indica was extracted. Ethanol extract was characterized by Gas Chromatography- Mass Spectroscopy. Seven ...
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PHYTOCHEMICAL ANALYSIS AND ANTITUBERCULAR ACTIVITY OF CENTRATHERUM ANTHELMINTICM SEED EXTRACT
... ABSTRACT: About 4 extracts (hexane, acetone, ethanol, and methanol extraction) from the seeds of Centratherum anthelminticum was extracted. Gas Chromatography-Mass Spectroscopy characterized ethanol extract. Seven ...
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Evaluation of Antimicrobial and Antitubercular Activity of 5-Nitro 2-Thiophene Carboxaldehyde by Invitro Method.
... antibacterial activity was carried out for 5-Nitro 2-Thiophene carboxaldehyde compound using Agar well diffusion method against Staphylococcus aureus, Enterococcus, ...antibacterial activity on Agar ...
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Synthesis and Antitubercular Activity of N3,N5-Diaryl-4-(5-arylisoxazol-3-yl)-1,4-dihydropyridine-
... This work was supported by grants from Research Council of Tehran University of medical Sciences and INSF (Iran National Science Foundation). We are thankful of TAACF (Tuberculosis Antimicrobial Acquisition & ...
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Synthesis, characterization and evaluation of antitubercular and analgesic activity of some novel pyrazolopyrimidine and pyrazolopyridine derivatives
... Desired fused ring system4{1.phenyl-3(Substituted phenyl)-1H-pyrazole-4-yl}-6-phenyl-1,2,3,4 tetrahydro pyrimidine-2thione & 5-phenyl –s-triazolo[ 1,5,a]pyrimidine (5,a,b) have been synthesized respectively with ...
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Synthesis, SAR study and evaluation of mannich and schiff bases of pyrazol-5(4H)-one moiety containing 3-(hydrazinyl)-2-phenylquinazolin-4(3H)-one
... vitro antitubercular potential of synthesized Mannich and Schiff bases was determined against ...of antitubercular activity (Table 5) indicated that varying degree of antitubercular ...
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Design and synthesis of some new imidazole and 1,2,4-triazole substituted fluorobenzimidazoles for antitubercular and antifungal activity
... anti-tubercular activity and was synthesized to see its effect on activity ...antituberculosis activity with compounds bearing a benzyl group at 1 st position ...the antitubercular ...
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SYNTHESIS AND EVALUATION OF ANTITUBERCULAR AND ANTI FUNGAL ACTIVITY OF SOME NOVEL 6 (4 SUBSTITUTED ARYL) 2 (3,5 DIMETHYL 1H PYRAZOL 1 YL) IMIDAZO[2,1 B] [1,3,4] THIADIAZOLE DERIVATIVES
... Antitubercular activity done against Mycobacterium tuberculosis of H37Rv Strain in BACTEC[15,16] medium using a broth micro dilution assay .The Microplate Alamar Blue Assay (MABA)[8] Compounds exhibiting ...
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Synthesis of novel phenyl azo chalcone derivatives for antitubercular, antiinflammatory and antioxidant activity
... The authors wish to thank Dr Shobha Rani RH, principal, Al-Ameen College of Pharmacy, Bangalore for encouraging and providing facility to carry out the research work. Mr Manish, Panjab University, Chandigarh for ...
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Design, Synthesis and Biological Evaluation of Novel Antitubercular Agents by Combining Pyrazoline and Benzoxazole Pharmacophores
... Jensen medium (L. J. medium) (Stover et al., 2000) [24] where the susceptibility of the compounds against multidrug-resistant TB (MDR-TB) and extensively drug-resistant TB (XDR-TB) strains were also checked. Eggs were ...
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“Isolation, Characterization of Bioactive Compounds and Evaluation of Anti-tubercular Activity of Ricinus communis Linn.” by Dr. Smt. Padma Ladda, Dr. Chandrakant Magdum, Dr. Mrs. Nilofar Naikwade, India.
... tubercular activity of plant and chemical constituents of leaves extracts of this ...anti-tubercular activity against ...the antitubercular activity of various bioactive compounds obtained ...
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