benzothiazole derivatives
Synthesis, Characterization and Drug-Likeness Predictions of 1,3-Thiazole and Benzothiazole Derivatives
... Heterocyclic compounds bearing nitrogen and sulphur in the main skeleton are reported to be a bioactive group. Thiazole and benzothiazole moieties are biologically significant class of this group. This research ...
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SYNTHESIS AND BIOLOGICAL EVALUATION OF SOME NEW BENZOTHIAZOLE DERIVATIVES
... amino benzothiazole derivatives: Take equimolar amount of substituted 2-hydrazinyl 1,3- benzothiazole derivatives and substituted acetophenone in methanol, add 2-4ml of formaldehyde and add ...
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A COMPREHENSIVE REVIEW ON BENZOTHIAZOLE DERIVATIVES FOR THEIR BIOLOGICAL ACTIVITIES
... Gupta and his colleagues designed a one-pot, solid phase, solvent-free microwave reaction which includes 2-aminothiophenol and various benzoic acid to synthesize various benzothiazole derivatives in a high ...
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Design Synthesis Characterization and Biological Evaluation of Some Novel Benzothiazole Derivatives as Anti Tubercular Agents Targeting Glutamine Synthetase 1
... NOVEL BENZOTHIAZOLE DERIVATIVES AS ANTI-TUBERCULAR AGENTS TARGETING GLUTAMINE SYNTHETASE 1” submitted by the candidate bearing the Register No:261515701 in partial fulfillment of the requirements for the ...
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BIOLOGICAL EVALUATION OF SOME SYNTHESIZED BENZOTHIAZOLE DERIVATIVES AND THEIR CHARACTERIZATION
... 3-benzothiazole derivatives are an important class of heterocyclic ...The benzothiazole nucleus containing compounds in this work is been treated with hydrazine hydrate to form hydrazone derivative ...
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SYNTHESIS, CHARACTERIZATION AND BIOLOGICAL INVESTIGATION OF SOME BENZOTHIAZOLE DERIVATIVES
... 13. Teenu James, Arya Rajendran, Shilpa Martin, Reshma Easo, Navneeth C. Krishnan, Asha Asokan Manakadan, Saranya TS., Computational approach on the drug affinity studies of substituted ...
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Antioxidant activity of novel coumarin substituted benzothiazole derivatives
... substituted derivatives of benzothiazole and they were evaluated for antioxidant activity by DPPH radical scavenging ...substituted benzothiazole derivatives showed significant antioxidant ...
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3D QSAR STUDY OF BENZOTHIAZOLE DERIVATIVES AS p56lck INHIBITORS
... ABSTRACT: 3D-QSAR models of Comparative of Molecular Field Analysis (CoMFA) and Comparative of Molecular Similarity Indices Analysis (CoMSIA) of 44 potent p56 lck inhibitors were performed. The conventional ligand-based ...
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Synthesis of some benzothiazole derivatives evaluated as antimicrobials and antibiofilms
... of benzothiazole derivatives, one incorporating the dihydropyrimidinone nucleus and the other one incorporating the 2-imino- thiazolidin-4-one structure hoping to obtain highly potent, more specific and ...
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RECENT ADVANCEMENT IN BIOLOGICAL APPLICATIONS OF BENZOTHIAZOLE DERIVATIVES: A SHORT REVIEW
... the benzothiazole nucleus found to play an important role as antimicrobial, anti-inflammatory, anticancer and antidiabetic ...fluoro- benzothiazole derivatives and then followed by screening for ...
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Synthesis and Biological Evaluation of 2-Phenyl Benzothiazole Derivatives as Cytotoxic Agents
... 2-phenyl benzothiazole derivatives was synthesized, biologically evaluated against breast cancer cell line (T47D) and compared with etoposide as a reference ...
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A theoretical evaluation on benzothiazole derivatives as corrosion inhibitors on mild Steel
... Benzothiazole derivatives have been studied extensively for their diverse chemical reactivity and potential broad spectrum of biological ...discovery. Benzothiazole moieties are part of compounds ...
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COMMON METHODS TO SYNTHESIZE BENZOTHIAZOLE DERIVATIVES AND THEIR MEDICINAL SIGNIFICANCE: A REVIEW
... of benzothiazole is a considerable area of current .... Benzothiazole derivatives possess a wide spectrum of biological applications such as antitumor ...
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Benzothiazole derivatives substituted in position 2 as biologically active substances with plant growth regulation activity
... stituted benzothiazole derivatives also influenced growth in cucumber, wheat coleoptile, mung bean and buckwheat and may be characterized as biologi- cally active substances with dominant auxine-like growth ...
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Synthesis, Characterization and Antioxidant Activity of Novel 2 Aryl Benzothiazole Derivatives
... of benzothiazole derivatives were ...synthesized derivatives were characterized by ATIR and Proton Nuclear Magnetic Resonance ( 1 H-NMR) ...synthesized benzothiazole derivatives showed ...
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A review on Indole and Benzothiazole derivatives its importance
... of benzothiazole based anti-inflammatory agents have been synthesized ...2-amino benzothiazole derivatives and evaluated them for anti- inflammatory ...amino benzothiazole is substituted at 4 ...
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Synthesis and antibacterial activity of new complexes of benzothiazole derivatives
... 2-amino benzothiazole were intensively studied as central muscle ...aromatic benzothiazole[15] nucleus is associated with variety of antihistamine activity, pharmacological activities,[9,10] such as ...
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SYNTHESIS, CHARACTERIZATION AND PHARMACOLOGICAL STUDIES OF BIOLOGICALLY ACTIVE BENZOTHIAZOLE DERIVATIVES
... of benzothiazole have been of great interest to medicinal chemistry [1], because its derivatives possessed various biological activities [2] such as anticancer [3-5], antihypertensive [6], antimicrobial ...
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SYNTHESIS AND ANTIBACTERIAL EVALUATION OF BENZOTHIAZOLE DERIVATIVES
... newer derivatives of benzothiazole with enhance antibacterial ...different derivatives were synthesized. The synthesized derivatives showed very good antibacterial activities against ...
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The effect of some benzothiazole derivatives as antioxidants for base stock
... requirements the lowest possible level of sulfur and phosphorus content of any additive has to be used in the formulation of industrial oil (4,5). It is well known that most of heterocyclic compounds which have compact ...
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