benzoxazole derivative
Synthesis and antimicrobial activity of some 2 phenyl benzoxazole derivatives
... to benzoxazole derivatives and have prompted researches around the globe to synthesize and explore the wide applicability of this important pharmacophoric ...
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Design, Synthesis and Antimicrobial Evaluation of Novel Benzoxazole Derivatives [Retracted]
... with benzoxazole skeletons that displayed potential antimicrobial activities ...of benzoxazole derivatives has been developed, some of which have exerted good minimum inhibitory concentration (MIC) values ...
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Design, Synthesis, Characterization And Evaluation Of Benzoxazole Derivatives For Their Antihyperglycaemic Activity
... substituted benzoxazole as a lipophilic tail, 2,4-thiazolidinedione as an acidic head and no carbon chain as a ...like benzoxazole, 2,4-thiazolidinediones and aromatic thioethereal alkyl group as central ...
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Synthesis of some benzoxazole derivatives and their anti inflammatory evaluation
... of benzoxazole derivatives throughthe reaction of substituted 2-aminophenols and acyl chlorides in the presence ofcatalytic amount of In(OTf)3 under solvent-free reaction ...2-substitued benzoxazole in good ...
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Synthesis and in vitro antitumor activity of new benzothiazole and benzoxazole derivatives
... A series of benzothiazole and benzoxazole derivatives were synthesized from their parents whom bearing o- aminocyano groups then functionalized on amino group or cyano group. Some of the newly formed compounds ...
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Design, synthesis and biological evaluation of benzoxazole derivatives as cyclooxygenase inhibitors
... 3-aminoalkyl-2-oxo-3H- benzoxazole derivatives also demonstrated potent analgesic and anti-inflammatory activity, and showed that these compounds exerted their in vivo activity by inhibiting the synthesis of ...
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Synthesis and invitro evaluation of novel benzoxazole derivatives as specific cyclooxygenase – 2 inhibitors
... 2-(2-chloroacetamido) benzoxazole-5-carboxylate with different secondary amines to give the corresponding methyl 2- {(2-dialkylamino) acetamido)}-benzoxazole-5-carboxylates (VIIa - ...the benzoxazole ...
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SYNTHESIS, CHARACTERIZATION AND ANTI MICROBIAL ACTIVITY OF SUBSTITUTED BENZOXAZOLE DERIVATIVES
... novel benzoxazole compounds were synthesized and evaluated for anti-microbial ...substituted benzoxazole with oxalic acid,cinnamicacid, succinic acid,phthalic acid,salicylic ...
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Synthesis of some novel benzoxazole derivatives and their antimicrobial activity
... The novel pyrazole derivatives were synthesized by means of cyclization reaction between equimolar quantities of substituted chalcone intermediates (0.02 mol) and hydrazine[r] ...
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Benzoxazole derivatives: design, synthesis and biological evaluation
... The method to synthesize the designed benzo- xazole derivatives is given in Scheme 1. Initially, 2-(chloromethyl)-1H-benzo[d]imidazole (I) was syn- thesized by the reaction of ortho phenylenediamine, chloroacetic acid ...
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Synthesis, characterization, and anticancer activity of benzoxazole derivatives
... So further molecular modification is required in order to arrive at more accurate structure activity relationship with their anticancer activity on breast cancer cell lines or different [r] ...
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Synthesis, characterization and biological evaluation of benzoxazole derivatives
... containing benzoxazole moiety, either isolated from plants or accessed by total synthesis, have remarkable biological activities [3] like antimicrobial [4] , antihistaminic [5] , antiparasitics [6] ,antiviral [7] ...
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5 Iodo 3 phenyl 2,1 benzoxazole
... in the asymmetric part (A and B), see Fig. 1. The molecules are almost planar, the dihedral angles between the mean planes of benzoisoxazole and benzene rings being 4.2 (3)° and 4.1 (3)° for A and B, respectively. The ...
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Benzoxazole: The Nucleus of Diverse Biological Activities
... 3-aminoalkyl-2-oxo-3H- benzoxazole derivatives also demonstrated potent analgesic and anti-inflammatory Activity, and showed that these compounds exerted their in vivo activity by inhibiting the synthesis of ...
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Benzoxazole: The molecule of diverse biological activities
... H. Ozan Gulcan et al (20) synthesized 4-(5-chloro-2-oxo-3H-benzoxazol-3-yl) butanamide derivatives and were screened for their analgesic and anti-inflammatory activities 15 as well as gastric ulceration potential in ...
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3 Benzyl 5 methyl 1,2 benzoxazole 2 oxide
... Benzoxazole derivatives show antiepileptic, antispasmodic and antifungal properties (Jian et al., 2007). 3-substituted 1,2- benzisoxazole derivatives are emerging as potential antipsychotic compounds, antiseizure ...
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2 (4 Aminophenyl) 1,3 benzoxazole
... The benzoxazole rings sytem is one of the most common heterocycles in medicinal ...new benzoxazole derivatives, and we report the crystal stucture ...
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SYNTHESIS, CHARACTERIZATION AND ANTI BACTERIAL ACTIVITY OF NOVEL 2-MERCAPTOBENZOXAZOLE DERIVATIVES Narender Boggula*, Ridhika M Patel, Akhil Rapolu, Pramod Kumar Bandari, Krishna Mohan ChinnalaDOWNLOAD/VIEW
... active benzoxazole derivatives have been known for long time, since they are the isosteres of naturally occurring cyclic nucleotides and they may easily interact with the biopolymers of the ...
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SYNTHESIS, CHARACTERIZATION AND EVALUATION OF IN VITRO CYTOTOXIC, ANTIBACTERIAL, ANTIOXIDANT ACTIVITY AND MOLECULAR DOCKING STUDIES OF NITRO SUBSTITUTED BENZOXAZOLE LINKED THIAZOLIDINE DERIVATIVES
... of benzoxazole with thiazolidine derivatives were synthesized by the cyclization of substituted Schiff’s base with thioglycolic ...synthesized benzoxazole with thiazolidine derivatives 6(a-j) exhibited ...
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ANTI FUNGAL AND ANTI OXIDANT ACTIVITIES OF NOVEL 2-MERCAPTOBENZOXAZOLE DERIVATIVES
... benzimidazole, benzoxazole, have been studied and found to be possessing interesting pharmacological ...active benzoxazole derivatives have been known for long time, since they are the isosteres of ...
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