Synthesis and activities
SYNTHESIS OF PYRAZOLE DERIVATIVES AND THEIR ANTIMICROBIAL ACTIVITIES
... CONCLUSION This study reports the successful synthesis of the title compounds in good yields and shows measurable antimicrobial activities. The present method is efficient, mild, simple, convenient and ...
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SYNTHESIS AND BIOLOGICAL ACTIVITIES OF FUSED HETEROARYLS
... anticancer activities, 12 and inhibitory of HIV-1 protease. 13 The synthesis of coumarins by the condensation of phenols and ethyl acetoacetate via Pechmann condensation in the presence of catalysts like ...
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Synthesis and antimicrobial activities of substituted phenylthioureas
... antibacterial activities and antifungal activities _____________________________________________________________________________________________ INTRODUCTION A review of the literature reveals that number ...
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Synthesis and biological activities of quassinoid analogues
... Chapter 3 - Z/t Vitro antimalarial Activities of Quassinoid Analogues 3.1 Introduction Plants have been an important source of clinical agents in the past and have considerable potential as sources of new drugs. ...
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Synthesis, anticancer and antioxidant activities of 6,8 dibromoflavones
... permits activities higher than that of ...the synthesis of biologically active natural products such as vitexin (Frick et ...1933) synthesis via chalcones ) and synthesis via an intramolecular ...
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Flux Synthesis and Photocatalytic Activities of Metal Oxides.
... during synthesis, contrasting particle morphologies can be obtained that also affect the photocatalytic ...photocatalytic activities of nearly four times greater than their platelet-structured ...
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Synthesis and Antiproliferative Activities of Triphenylmethanol Conjugates of Leuprorelin
... the synthesis of the antioxidant tri- phenylmethanol (TPMs) derivatives of LEP through the covalent conjugation with dodecanedioic acid as the ...antiproliferative activities in multiple cell ...
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Synthesis, antimicrobial, and antiproliferative activities of substituted phenylfuranylnicotinamidines
... the synthesis of a series of substituted phenylfuranylnicotinamidines using facile syn- thesis ...biological activities of this class led to discovery of their anticancer, antimicrobial, DNA cleavage, and ...
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Synthesis and antioxidant activities of hydroxylated coumarinyl chalcones
... iv ABSTRACT Hydroxylated coumarins and chalcones are known to possess potent antioxidant activities. The present study highlights the synthesis of two hydroxycoumarins namely 3-acetyl-7-hydroxycoumarin and ...
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Synthesis of Substituted Chalcones and Investigation of Their Biological Activities
... The synthesis of highly antioxidants and antimicrobial agents has attracted great attention due to their high importance to human ...biological activities such as anticancer, antibacterial and ...
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Synthesis and antimicrobial activities of 9H-carbazole derivatives
... promising activities against some tested microorganisms which may be due to the increase the lipophilic character of the mol- ecules, which facilitate the crossing through the biological membrane of the ...
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Synthesis of cinnamamide derivatives and their α-glucosidase inhibitory activities
... DISCUSSION SYNTHESIS OF CINNAMAMIDE DERIVATIVES Synthetic cinnamamide derivatives were synthesized and assayed for their α-glucosidase inhibitory activities (Scheme 1 and Table ...
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SYNTHESIS & ANTIMICROBIAL ACTIVITIES OF HYDRAZO METAL COMPLEX LIGANDS
... These complexes also perturb the respiration process of the cell and thus block the synthesis of the proteins that restricts further growth of the organism. In addition to this, many other factors, such as ...
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Synthesis and antibacterial activities of enamine derivatives of dehydroacetic acid
... the synthesis of dehydroacetic acid (1) from N-hydroxysuccinimdyl acetoacetate, a novel series of enamine-based derivatives were synthesised in order to improve the antibacterial activity of dehydroacetic ...
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NOVEL SYNTHESIS AND ANTIMICROBIAL ACTIVITIES OF THIAZINO-OXAZINE DERIVATIVES
... Novel Synthesis and Antimicrobial Activities of Thiazino-Oxazine Derivatives Pravina B. Piste * P. G. Department of Chemistry, Yashavantrao Chavan Institute of Science, Satara-415001, Maharashtra, India ...
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Synthesis and Characterization and Biological Activities of Hydrazones
... ABSTRACT: Hydrazones derivatives of carbonyl compounds constitute an important class of biologically active compounds. Metal complexes of Schiff bases represent an important class of coordination compounds. Schiffs base ...
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The synthesis of novel pyrophosphate analogues and their antiviral activities
... 1.5 Outline of Work Undertaken The aim of the present work was to investigate the preparation of novel substituted methylenebisphosphonates and to examine the activities of a broad range of these compounds against ...
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Synthesis and Anti Cancer Activities of Resveratrol Derivatives
... et al. [19] tested the activity of 70 different resveratrol analogues as aromatase for chemotherapy cancer. The aromatase inhibitory activities of some analogues were much more effective than the lead compound ...
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Synthesis and Biological Activities of [1,3] Oxazine Derivatives
... General method for synthesis of substituted 4 (a-f) Equimolar quantity of N-(4-Acetylphenyl)-nicotinamide (0.01 mol) and substituted benzaldehyde (0.01 mol) were dissolved in absolute alcohol and 40% KOH solution ...
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Synthesis and Biological Activities of Some Benzodiazepine Derivatives
... chemical synthesis techniques we have used catalysts which have shown catalytic activity for chalcone and have many advantages over catalyst like NaOH, KOH such as ease of handling, low cost and elimination of ...
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