THIAZOLE DERIVATIVES
Synthesis of some novel thiazole derivatives
... Thiazoles are important class of heterocyclic compounds, found in many potent biologically active molecules such as sulfathiazole (antimicrobial drug), Ritonavir (antiretroviral drug), Abafungin (antifungal drug) ...
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New thiopyrano[2,3-d][1,3]thiazole derivatives as potential antiviral agents
... The screening of 24 thiopyrano[2,3-d][1,3] thiazole derivatives against a wide range of viru- ses has been carried out. Some compounds possess mode rate levels of the antiviral activity. However, the ...
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Synthesis and characterization of novel thiazole derivatives of disubstituted N arylmaleimides
... General procedure for the preparation of thiazole derivatives of Disubstituted N- aryl maleimides: (7a-g) The thiosemicarbazone 5(0.01 mol) in ethanol (10 mL) was stirred for 10 min. To this mixture ...
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Syntheses and antimicrobial activity of some new thiohydantoin and thiazole derivatives
... The researches study the successful synthesis and antimicrobial activity of some new thiohydantoin , thiazole derivatives .The investigation of antifungal and antibacterial activity data revealed that all ...
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INHIBITION OF SPLEEN TYROSINE KINASE (SYK) IN SILICO BY THIAZOLE DERIVATIVES
... thiazoles derivatives showed wide range of biological ...substituted thiazole containing derivatives as SYK inhibitor was ...substituted thiazole containing ...the thiazole ...
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Synthesis and antimicrobial activity of some novel 2 amino thiazole derivatives
... Thiazole derivatives are an important class of heterocyclic ...their derivatives have attracted continuing interest over the years because of their varied biological ...activities. Thiazole, ...
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DESIGN, SYNTHESIS, AND PHARMACOLOGICAL EVALUATION OF SOME NOVEL BIS THIAZOLE DERIVATIVES
... Heterocyclic chemistry is now fast-growing research field in chemistry. Thiazoles are five-membered heterocycles with N and S as a heteroatom. They are ubiquitous in natural product [1] and pharmaceuticals [2]. ...
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Antibacterial Effects of Novel Thiazole Derivatives and the Toxicity of Oxothiazole on Liver Histopathology of Mice
... of thiazole derivatives which their results indicated to the compounds inhibitory action with halo diameter of ...these derivatives on gram positive Staphylococcus aureus is lesser than our ...the ...
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Effect of Thiazole Derivatives on the Corrosion of Mild Steel in 1 M HCl Solution
... many thiazole derivatives have been studied as corrosion inhibitors and found that thiazole derivatives have good corrosion inhibition effect ...of thiazole compounds is attributed to ...
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SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL 1, 3 THIAZOLE DERIVATIVES
... The introduction of a variety of antibacterial agents in multiple unrelated drug classes, resistance continues to emerge. The pharmaceutical researcher must respond to these clinical challenges by bringing forward a ...
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SYNTHESIS AND CHARACTERIZATION OF NOVEL ADAMANTANE BASED THIAZOLE DERIVATIVES AS POTENTIAL ANTIBACTERIAL AGENTS
... Adamantane based thiazole derivatives and its derivatives are very well known in medicinal and agricultural chemistry [1]. Among the various classes of heterocyclic compounds, thiazoles are ...
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Synthesis Characterization and antitumor activity of thiazole derivatives containing indole moiety bearing-tetrazole
... of thiazole derivatives containing Indole moiety bearing tetrazole ring were synthesised by the condensation of 2-(3-(3chloro -1-(4-substitued phenyl )-tetrazole -2-yl(1H-Indole –yl Aceto hydrazone with ...
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A facile synthesis, and antimicrobial and anticancer activities of some pyridines, thioamides, thiazole, urea, quinazoline, β-naphthyl carbamate, and pyrano[2,3-d]thiazole derivatives
... gyrase B [25]. In addition, pyrano[2,3-d]thiazoles are biologically interesting compounds with diabetes, obe- sity, hyperlipidemia, and atherosclerotic diseases [26]. They are also known to show antimicrobial, bacteri- ...
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Effective Protection for Copper Corrosion by Two Thiazole Derivatives in Neutral Chloride Media: Experimental and Computational Study
... its derivatives are the most successful series due to the high performance and low ...Many thiazole derivatives are explored as corrosion inhibitors for mild steel [29-32], and few of them have been ...
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Stereoselective synthesis, X-ray analysis, computational studies and biological evaluation of new thiazole derivatives as potential anticancer agents
... different thiazole derivatives has attracted great attention due to their diverse biological activities that include anticonvulsant [1, 2], antimicrobial [3, 4], anti-inflammatory [5, 6], anticancer [7], ...
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Electrochemical and Quantum Chemical Studies on Adsorption and Corrosion Inhibition Performance of Quinoline -Thiazole Derivatives on Mild Steel in Hydrochloric Acid Solution
... quinoline-thiazole derivatives namely, {4-[1-aza-2-(phenyl)vinyl]-3-phenyl-2- thioxo(1,3-thiazoline-5-yl)}-N-[1-aza-2-(2-chloro(3-quinolyl))vinyl] (Inh I) and {4-[1-aza-2-(4- ...
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Effect of Thiazole Derivatives on Copper Corrosion in Acidic Sulphate Solution
... inhibitors are lower than that obtained in the inhibitor free solution and decrease uniformly with the increase of inhibitors concentration. This reduction of the activation energy in the presence of thiazole ...
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REVIEW: SYNTHESIS SCHEMES OF ANTIMICROBIAL AND ANTICANCER THIAZOLE DERIVATIVES
... compounds. Thiazole derivatives are an important class of heterocyclic ...their derivatives have attracted continuing interest over the years because of their varied biological activities and are ...
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SYNTHESIS AND ANTI INFLAMMATORY ACTIVITY OF THIAZOLE DERIVATIVES
... of thiazole derivatives is important for their wide range of pharmaceutical and biological .... Thiazole derivatives display a wide range of biological activities such as cardiotonic, ...
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Synthesis and Biological Evaluation of Isatin Based Thiazole Derivatives
... their derivatives particularly in medicinal fields, because isatin plays a key effect like ascorbic acid, hydroxyl amino acids, omeprazole, thiol compounds and imidazole ...
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