[PDF] Top 20 Syntheses and antitumor activity of some 1,2,4 - triazine derivatives
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Syntheses and antitumor activity of some 1,2,4 - triazine derivatives
... and antitumor activities of the synthesized compounds 3-7 were tested against the HCT-116 cell line according to method of Mossman [15], Gandadevi and Muthumary ... See full document
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SYNTHESIS, CHARACTERIZATION AND PHARMACOLOGICAL EVALUATION OF SOME NEW 6 (3,5 SUBSTITUTED 2 BROMO/HYDROXY PHENYL) 1,2,4 TRIAZINE DERIVATIVES AS ANTICONVULSANT AGENTS
... 6-(3,5-Substituted-2-bromophenyl)-1,2,4-triazine derivatives and 6-(3,5- substituted-2-hydroxyphenyl)-1,2,4-triazine derivatives were prepared from 6-(2- ... See full document
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Biological activity and mass spectra investigation of synthesized 1, 2, 4 triazine derivatives
... 1, 2, 4-Triazine derivatives (3, b) were prepared via condensation of oxazolinones (2a, b) with thiosemicarbazide in acetic ...[2,1-a]-1,2,4-triazine derivatives (6 and ... See full document
12
Syntheses, characterization and antimicrobial screening of some novel 3, 5 diaryl 4H 1, 2, 4 triazole derivatives
... The syntheses of a series of 3, 5-diaryl-4H-1, 2, 4-triazole derivatives are ...antibacterial activity against ...the 1, 2, 4- triazole moiety at position ... See full document
5
SYNTHESIS, SPECTRAL AND BIOLOGICAL STUDIES OF SOME s TRIAZINE DERIVATIVES OF 1 (1 (4METHXYPHENYL)ETHYL) CYCLOHEXANOL
... phenyl)-1,3,5-triazin-2-amine with 1-(2-amino-1-(4-methoxyphenyl)ethyl)cyclohexanol. Products of step-II (a1 to a10) were taken in 80 ml acetone in an RBF and added ... See full document
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Synthesis, Characterization and Antitumor Activity of Some Novel Pyrimidine Sulfonamide Derivatives
... pyrimidine derivatives incorporating sulfonamide moiety such as: imidazopyrimidine 3a,b, pyrimidoquinazoline 4a,b and pyrimidothiazine derivatives 5a,b, respectively, in good ...S-Methylpyrimidine ... See full document
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Synthesis, characterization and antimicrobial activity of some novel s triazine derivatives incorporating quinoline moiety
... Bi substituted cyanuricchloride 3.8g(0.01mol) was added slowly to N 1 –(7-chloro quinoline -4-yl) ethane-1,2 – diamine.2.21g(0.01mol) in acetone (35ml) with constant stirring for 6hr above 60°c. sodium ... See full document
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Synthesis and evaluation of antioxidant and antitumor activity of some heterocyclic benzocoumarin derivatives
... : 1-[(Bezocoumarin-3-ylethylidene)amino]-thiourea (2) was prepared via condensation of 3-acetyl benzocoumarin (1) with thiosemicarbazide, Reaction of compound 2 with acetic anhydride and ethyl ... See full document
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SYNTHESIS, SPECTRAL AND BIOLOGICAL EVOLUTION OF 2 (4 FLUOROPHENYL 1, 3, 4 OXADIAZOL 2 –YL 5 SULFANYL) 4 (CYCLOHEXYLAMINO) 6 (ARYLAMINO) S TRIAZINE
... their derivatives are important intermediates in organic synthesis and widespread application in medical ...s- triazine derivatives were synthesised with different substituted aryl ...synthesis ... See full document
5
Syntheses and antibacterial activity of some 1 phenyl 3 (4 (4 butanoloxy) phenyl) 5 aryl 1H pyrazoles
... pyrazole derivatives as a source of new antibacterial agents. Pyrazole derivatives have been reported to possess diverse biological activities such as antimicrobial [2], antibacterial [3-6], ... See full document
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Synthesis, Molecular Docking and evaluation of Antiangiogenic activity and Cellular metastasis potential of some Triazine and Pyrrolidin 2 one derivatives
... Table 1. The syntheses of triazine and pyrrodine-2-one derivatives (2a-2h and 4a-4d) are outlined in scheme 1 and ...amino-1,2,4 triazine or pyrrodine-2-one ... See full document
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Syntheses and antimicrobial activity of some new thiohydantoin and thiazole derivatives
... acetyl derivatives (4 and 7). Reaction of 2-thiohydantoin (6) with thiophene-2-carboxaldhyde and chloroacetic acid gives 5-(thiophen-2-ylidene)-3-[(p-tolylethylidene)amino] -2- ... See full document
6
Synthesis of Some Novel Quinazolino-Triazine Derivatives for Their Antimicrobial Activity
... antibacterial 1 , analgesic 2 , anti- inflammatory 3 , antifungal 4 , antimalarial 5 , antihypertensive 6 , CNS depressant 7 , anticonvulsant 8 , antihistaminic, local anaesthetic 9 , ... See full document
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Formulation and Antibacterial Evaluation of Some Novel S-Triazine Based Chalcones and Their Derivatives
... chalcones, 2-(4'-chlorophenylamino)-4-(4'-flurophenylamino)-6-[4'-3{3"- (substituted phenyl/2-thienyl/2furanyl)-2"-propenon-1"-yl} ... See full document
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Synthesis and Antimicrobial Activity of 1 (4 aryl 2 thiazolyl) and 1 (4 aryl 2 oxazolyl) 3,5 diaryl 2 pyrazoline derivatives
... [8,9], antitumor [10] ,antidepressant [11], and antidiabetic [12], and since the combat against bacterial infections has resulted in the development of a wide variety of antibiotics, therefore, recent efforts have ... See full document
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Computation of Structure Activity and Design of Chalcone Derivatives
... chalcone derivatives were synthesized according to their physiological activities, such as anti-inflammatory [1], antiviral [2], antitumor [3], anticancer [4] and so ...chalcone ... See full document
8
Synthesis, Characterization and Anticonvulsant Activity of Some Novel 4, 5-Disubstituted-1, 2, 4-Triazole Derivatives
... novel 4, 5-disubstituted-1,2,4-triazoles (6a-o) were synthesized on refluxing hydrazinecarbothiomides with an aqueous solution of sodium hydroxide starting from methyl-4-hydroxy benzoate via synthesis of an ... See full document
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SYNTHESIS, CHARACTERIZATION AND ANTIMICROBIAL ACTIVITY OF SOME NEW 2-THIOXOIMIDAZOLIDIN-4-ONE DERIVATIVES
... Synthesis of (E)-2-phenyl-1-(1- phenylethylidene)hydrazine:To a methanolic solution of acetophenone(0.01M) and phenyl hydrazine(0.01M), small amount of concentrated hydrochloric acid was added and ... See full document
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SYNTHESIS, CHARACTERIZATION AND ANTIMICROBIAL ACTIVITY OF SOME NEWLY 1, 2, 4 TRIAZOLE DERIVATIVES
... Medicine 2 , LLRM Medical College, Meerut - 250002, Uttar Pradesh, ...of 1-(2-(4H-1,2,4-triazol-4-yl)ethylamino)-3-ch- loro-4-(5-methoxy/ehthoxy-2-substituted ... See full document
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A novel class of fluorinated A2A adenosine receptor agonist with application to last step enzymatic [18F]fluorination for PET imaging
... The formation of alkyne 18 was achieved from commercially available N-Boc-4-piperidinemethanol 14. Introduction of a tosyl group to N-Boc-4-piperidinemethanol 14 afforded 15 which, after flash ... See full document
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