QUINOLINE DERIVATIVES
Synthesis and biological screening of some novel Quinoline derivatives
... of quinoline derivatives 2-chloro 3-formyl quinoline, 3-chloro-4(2- chloroquinolin-3-yl)1-phenyl amine azetidin 2-one, 3-chloro-4(2-chloroquinolin-3-yl)2,4- dinitro phenyl amine azetidin 2-one, ...
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Chitosan decorated copper nanoparticles as efficient catalyst for one-pot multicomponent green synthesis of novel quinoline derivatives
... of quinoline derivatives via four- component one-pot reaction of P-Chlorobenzaldehyde, dimedone, ethyl cyanoacetate and ammonium acetate as the model reaction under ultrasound irradiation and its behavior ...
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THERAPEUTIC SIGNIFICANCE OF QUINOLINE DERIVATIVES AS ANTIMICROBIAL AGENTS
... antibiotics. Quinoline derivatives have proved their medicinal importance by having broad spectrum of pharmacological activities like antimicrobial, anticancer, antiviral and anti-inflammatory activities ...
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SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF SOME QUINOLINE DERIVATIVES
... INTRODUCTION: Quinoline derivatives represent one of the most active classes of compounds possessing a wide spectrum of biological ...of quinoline derivatives including their antimicrobial ...
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SYNTHESIS DOCKING AND QSAR STUDIES OF QUINOLINE DERIVATIVES
... Five novel quinoline derivatives were synthesized, characterized by IR spectroscopy, docking QSAR studies were performed for the designed compounds. For BPM-1 and BPM- 2 DOKING and QSAR studies revealed ...
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DIFFERENT QUINOLINE DERIVATIVES BY MICROWAVE IRRADIATION METHOD
... like quinoline alkaloids, therapeutics and synthetic analogues with very important biological activities such as antimalarial, antiasthmatic, antidiabetic, antibacterial, antiviral, anti-inflammatory, ...
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Synthesis and Pharmacological Evaluation of Some Quinoline Derivatives as Potential Antiamnesic Agents
... A deÞ cit of cholinergic neurotransmission is considered to be one of the major causes of disturbance in learning and memory. Among the various therapeutic approaches investigated to enhance cholinergic transmission, ...
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Biological evaluation of some quinoline derivatives
... Some new quinoline derivatives viz., benzodiazepines and aminopyrimidine were synthesized and their characterization was done by spectral data of IR, NMR and mass. The antibacterial activities were studied ...
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Chitosan decorated copper nanoparticles as efficient catalyst for synthesis of novel quinoline derivatives
... nanoparticles [39]. All of these catalysts showed pronounced catalytic activity due to their nanosized and large surface area features. In contrary to that the produced % yield of products especially after re-use of ...
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THIADIAZOLE-QUINOLINE DERIVATIVES AS POTENTIAL WOUND HEALING ACTIVITY
... of Quinoline derivatives is well known from many years ...various derivatives of quinolines are used to treat malaria (Vlabhov R et ...Furthermore quinoline compounds can possess ...
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SYNTHYSES, REACTIONAND CHARACTRIZATION OF QUINOLINE DERIVATIVES
... of quinoline derivatives starting with 4, 7- dichloroquinoline ...dithioacetal derivatives gave pyrazole derivatives 2a, b, respectively following Afred Kreutzberger et al [17, 18] ...
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Synthesis and molecular modeling of new quinoline derivatives as antitumor agents
... active quinoline analog that showed promising cytotoxic activity against the tumor cell lines and in agreement with the docking study results that indicated its favorable complementarity with the binding ...
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Design New Pyrano Quinoline Derivatives and Study of their Anti-Microbial Activity
... of derivatives having linkers of iminoether 2 position of benzo[h][1,6]naphthyridines In view of all these facts and as the continuation of our work on the synthesis of new heterocyclic derivatives by using ...
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Corrosion Inhibition of Carbon Steel by Lepidine in HCl Solution
... literature, quinoline and its derivatives have been investigated as corrosion inhibitors for many commercial metals because of the p-π conjugation of the quinoline ...of quinoline ...
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Antioxidant activity of alkoxy derivatives of (quinoline-4-ylthio)carboxylic acids
... Studying of quinoline derivatives acute toxicity showed that their DL 50 are 930 mg/kg and higher. It allows to consider these compounds as low-toxic or nontoxic substances (IV and V toxicity classes re- ...
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Quinoline and its Derivatives as Effective Corrosion Inhibitors for Mild Steel in Acidic Medium
... The importance of temperature variation in corrosion studies involving the use of inhibitors is to determine the mode of inhibitor adsorption on the metal surface [55, 56]. The influence of temperature on the corrosion ...
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Synthesis and Characterization of some New 6-substituted-2, 4-di (hetar-2-yl) Quinolines via Micheal Addition - Ring closure Reaction of Schiff base N-(hetar-2- yl) methylene aniline with Hetarylketones
... substituted quinoline derivatives via the reaction of aniline and hetarylchalcone analogues, despite the practical shortcomings the optimum condition was achived in two steps from the reaction of aniline ...
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Synthesis, Characterization and Catalytic Application of V2O5/Fe3O4 as Heterogeneous Catalyst for the Synthesis of Quinoline 4 carboxylic Acid Derivatives
... Quinoline derivatives were broadly studied because of their effective pharmacological and biological ...activities. Quinoline derivatives are widely used as antagonists [11], antitumour, ...
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Synthesis of Quinoline Containing Pyrazolone Derivatives and their Biological Studies
... compounds quinoline derivatives are known to contribute to various pharmacological ...the quinoline nucleus found in several natural products shows a varied biological ...The derivatives of ...
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SYNTHESIS, CHARACTERIZATION AND ANTIMICROBIAL ACTIVITY OF SOME NOVEL QUINOLINE BASED IMIDAZOLES
... imidazole derivatives have wide range applications in coordination chemistry 4 , organometallic catalysis 5 and asymmetric catalysis 6 ...synthesis. Quinoline moiety is present in many classes of ...
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