synthesised compounds
Effect of novel phenothiazine derivatives on brain dopamine in Wistar rats
... These compounds were prepared by modifications of the existing phenothia- zine by performing (1) a new substitute at nitrogen element in phenothiazine ring and (2) an introduc- tion of a hetero-aromatic ...the ...
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Virtual Screening Identifies New Scaffolds for Testosterone 17β Dehydrogenase (NADP+) Inhibitor
... 6 compounds are biologically important molecules and possess desirable molecular properties for drug likeness except log P values of C3 and ...of compounds to improve their hydrophilicity and ...synthesized ...
5
1, 3, 4 Oxadiazole as antimicrobial agents: An overview
... (2010); synthesised some novel 2-substituted-5-[isopropylthiazole] clubbed 1,3,4-Oxadiazoles (Compound 5 and 6) and tested for antimicrobial activity by broth microdilution ...various synthesised ...
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Drug design, development and screening of pyrazolo pyridazine as potential agent for treatment of breast cancer
... The compounds were characterized by analytical techniques like TLC, UV, IR, NMR Spectral ...the synthesised compounds were checked for drug likeliness using QIKPROP software and found to be ...
6
Synthesis, spectral studies and antimicrobial studies of 7 [phenylamino] 5 methyl 1,4 diazepines and its derivatives
... were synthesised in good to excellent yield via cyclocondensation of 1-N (substituted phenyl carboxamido) propane-2-one with ethylene ...catalyst. Synthesised compounds were ecofriendly and ...
5
Synthesis and In Vitro Antioxidant Activity of New 3-Substituted-2-?Oxindole Derivatives
... newly synthesised compounds were determined by using open capillary tubes in scientific melting point apparatus and are ...the synthesised compounds were recorded on Bruker Avance 400 ...
6
Design, synthesis, conformational and molecular docking study of some novel acyl hydrazone based molecular hybrids as antimalarial and antimicrobial agents
... were synthesised by condensation of 1,4-dihy- dropyridin-4-yl-phenoxyacetohydrazides with differently substituted pyrazole ...the synthesised compounds were screened for their in vitro antimalarial ...
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Synthesis and invitro anticancer screening of some novel benzotriazole derivatives
... were synthesised and are evaluated for invitro anticancer ...hydrogen compounds were selected and are reacted with benzotriazole and formaldehyde; with the removal of water molecule the desired mannich ...
6
Synthesis, Characterization and Thermal Stability Study of New Heterocyclic Compounds Containing 1,2,3-Triazole and 1,3,4-Thiadiazole Rings
... of synthesised p-substituted phenyl azides and propiolic ...heterocyclic compounds containing 1,2,3-triazole and 1,3,4-thiadiazole ring combined in one molecule was synthesised via a condensation ...
7
ANTIOXIDANT ANALYSIS OF SYNTHESISED HYDRAZO METAL COMPLEX LIGANDS
... synthesized compounds were tested for anti-oxidant activities by DPPH ...assay. Synthesised compounds showed good activity both in DPPH Scavenging radical assay, where as other compounds ...
13
Synthesis Characterization and Antioxidant Activity of Ni (II) and Co (II) Quinoline Schiff Base
... newly synthesised compounds has been determined at a different concentration range by means of their interaction with the stable free radical 1,1-diphenyl-2-picryl hydrazyl (DPPH) on the basis of spectral ...
6
IN VITRO ANTHELMINTIC ACTIVITY OF 3 (3 CHLOROPHENYL) 5 PHENYL 4, 5 DIHYDRO 1,2 OXAZOLE DERIVATIVES
... The synthesised compounds tested for anthelmintic activity for this compounds were prepared at concentration of 20, 40, 80 mg/ml using saline 5% DMF solvents and compare the results with the standard ...
7
Functionalisation of MWCNTs with poly(lauryl acrylate) polymerised by Cu(0) mediated and RAFT methods
... aromatic compounds employ π-π stacking and hydrophobic interactions to bind to the surface of ...al. synthesised pyrene functionalised poly(methyl methacrylate) (PMMA) via RAFT (PMMA-b-pyrene) to achieve ...
26
Synthesis and antimalarial activity of some nitrogenous heterocyclic compounds
... Chloroquine (I.2a) is generally considered to be one of the most fascinating, useful and versatile antimalarial drugs developed during the modern era of synthetic organic chemistry.12 It was first prepared in 1934 by H. ...
231
Luminescent water dispersible microporous polymeric nanospheres
... PPDs synthesised in this work were all shown to be porous and demonstrated long-term stability in a range of organic ...nitroaromatic compounds with excellent detection ...
12
Evaluation of Anticorrosive Effect of Synthesised Carveol Derivatives on Steel in Hydrochloric Acid
... corrosiveness media such chemical cleaning and pickling generally used to remove mill scales (oxide scales) from the metallic surface [3]. Though the existing data show that organic compounds have good ...
13
In line Test of Synthesised Systems Exploiting Latency Analysis
... This paper details an analysis technique for identifying and quantifying these latent periods by modelling the flow of control through the system as a Markov chain, which takes into account branching and feedback in the ...
27
Design, Characterisation and Anticonvulsant Evaluation of Thienopyrimidinone Derivatives Synthesised by Green Chemistry
... Melting points were determined in open capillary tubes and are uncorrected. Formation of the compounds was checked by TLC on silica gel-G plates of 0.5 mm thickness and spots were located by iodine and UV light. ...
8
ANTIBACTERIAL ACTIVITY OF NEWLY SYNTHESISED PYRIDINYL COUMARIN DERIVATIVES
... parent compounds such as 3-bromoacetyl coumarin, 3-bromoacetyl 6- bromocoumarin and 3-bromoacetyl 6-chlorocoumarin were refluxed with ethyl and methyl isonicotinate and nicotinate in toluene to obtain twelve ...
10
DESIGN, SYNTHESIS AND EVALUATION OF SOME NOVEL {[(1HINDOL 4 YL)OXY]METHYL} 5 PHENYL 1,3,4 OXADIAZOLE DERIVATIVES AS POTENTIAL ANTIOXIDANT AGENTS
... are synthesised by the reaction of 2-[(1H-indol- 4-yl)oxy]acetohydrazide (2) with different aromatic aldehydes to form schiff’s bases (3) and the cyclization of the 2-[(1H-indol-4-yl)oxy]-N'- ...
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