Inclusion Complexes
FORMULATION AND CHARACTERISATION OF AZITHROMYCIN DIHYDRATE INCLUSION COMPLEXES USING DERIVATIVES OF b-CYCLODEXTRINS AS COMPLEXING AGENTS
... Azithromycin Inclusion complex was analyzed to find out whether the Inclusion complexes of various drug polymer ratios are crystalline or ...(Azithromycin inclusion complex with Sulfobutyl ...
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Enhancement of dissolution and bioavailability of poorly soluble Telmisartan:Designing modified cyclodextrin inclusion complexes
... an inclusion complex with telmisartan (TEL), a poorly soluble drug and its related effects on dissolution rate and relative ...Resulting complexes were characterized by differential scanning calorimetry, ...
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Melarsoprol cyclodextrin inclusion complexes as promising oral candidates for the treatment of human african trypanosomiasis
... cyclodextrin inclusion complexes can most easily be explained by the more controlled delivery of the trypanocidal drug to the brain following a sustained absorption from the gut compared with that of an ...
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Synthesis and Characterization of Host Guest Inclusion Complexes of Cyclodextrin Molecules with Theophylline by Diverse Methodologies
... host–guest inclusion complexes have been produced with medicinally important guest molecule theophylline within aqueous α-Cyclodextrin and ...for inclusion with Theophylline which include diversified ...
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Utility of Sulfobutyl Ether beta-Cyclodextrin Inclusion Complexes in Drug Delivery: A Review
... optimised inclusion complex can be an efficient strategy to increase the solubility of poorly soluble compounds and provide stability to a large number of active pharmaceutical ...SBE-β-CD inclusion ...
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Preparation, Characterization and Evaluation of Human Guarded Chlorpyrifos Urea Co-inclusion Complexes
... co- inclusion complexes of insecticide resulting in two- in-one product for agricultural use ...CHUCIC complexes were characterized by FTIR, DSC, XRD and 1 ...
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CHARACTERISATION OF INCLUSION COMPLEXES BETWEEN BIFONAZOLE AND DIFFERENT CYCLODEXTRINS IN SOLID AND SOLUTION STATE
... NMR spectroscopy has been recognized as an important tool for the interaction study of CD and pharmaceutical compounds in solution state. This technique also gives information on the topology of the interaction between ...
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Optimisation of β-cyclodextrin inclusion complexes with natural antimicrobial agents: thymol, carvacrol and linalool
... prepare inclusion complexes, however, large-scale production is limited due to the size of the reaction tanks required and wastewater disposal considerations (Hedges, ...
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Experimental, molecular docking investigations and bioavailability study on the inclusion complexes of finasteride and cyclodextrins
... CyDs inclusion complexes. All the inclusion formulations displayed a more rapid dissolution rate and extent of FIN than the free drug, with a significant improvement in FIN dissolution from both HP- ...
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PREPARATION AND EVALUATION OF INCLUSION COMPLEXES OF FELODIPINE
... β-CD.The inclusion complexes made with HP β-CD exhibited higher dissolution rate than β-CD at lower proportions, hence HP β-CD complex at the ratio of 1:1 was ...
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Inclusion complexes of Ketoprofen with beta-cyclodextrins: Oral pharmacokinetics of Ketoprofen in human
... the inclusion complex with βCD attained peak plasma level of ...the inclusion complex were decreased, compared to that of powder alone, which relates to rapid dissociation of the complex, following the ...
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Improvement of Solubility and Dissolution Properties of Clotrimazole by Solid Dispersions and Inclusion Complexes
... and inclusion complexes equivalent to 20 mg of CLOT was carried out with the USP II Dissolution Test Apparatus (paddle) (Pharma Test SP6-400, Hamburg, Germany) at ...
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Synthesis and Characterization of Hydroxypropyl α-Cyclodextrin Inclusion Complexes with Azo Dyes
... of cyclodextrin complexes with turmeric oleoresin. Food Chem, 114 (2), 459-465 (2009). 16. Badr-Eldin SM, Elkheshen SA & Ghorab MM, Inclusion complexes of tadalafil with natural and chemically ...
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PRECLINICAL PHARMACOKINETIC EVALUATION OF EFAVIRENZ βCD POLOXAMER 407 PVP K30 INCLUSION COMPLEXES
... K30 inclusion complexes could be compressed into tablets by both wet granulation and direct compression methods retaining their fast dissolution rate ...K30 inclusion complexes to assess their ...
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SYSTEMATIC OPTIMIZATION OF FORMULATION OF INCLUSION COMPLEXES CONTAINING AN ANTI DIABETIC DRUG
... Cyclodextrins (CDs) form a group of structurally related oligosaccharides with cylinder- shaped cavities that have the capacity to form inclusion complexes with many drugs by taking a whole drug molecule, ...
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Mosquito repellent activity of cotton functionalized with inclusion complexes of β-cyclodextrin citrate and essential oils
... natural repellents as essential oils are the upcoming genre of scientific interest due to their non-toxic, non-sticky, non-irritating and eco-friendly nature; however, essential oil repellents tend to being short-lived ...
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EFFECT OF PVA ON HP β- CD INCLUSION COMPLEXES OF DICLOFENAC FOR ENHANCING ITS DISSOLUTION RATE
... CD complexes followed first order ...the inclusion complexes. The dissolution data of all inclusion complexes prepared obeyed Hixson-Crowell’s cube root model indicating that the ...
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Electrochemical Evaluation of the Controlled Release Behaviors of the Cyclodextrin Inclusion Complexes on the Drug Deliveries to Microbial Cell
... In the literature, some CDs associated with biocides are described as active or inactive on bacterial growth [3]. As example, Schmidt et al. showed that encapsulated organic biocides are significantly more active than ...
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The Electrochemical Investigation of Inclusion Complexes of Nifedipine and Amlodipine with B-Cyclodextrin and (2-Hydroxypropyl)-B-Cyclodextrin
... It was observed that complexation with amlodipine and nifedipine in all the cases causes two main changes in cyclic voltammograms compared to their standards. Firstly, the initial potential of the anodic reaction as well ...
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Multifunctional dendrimer/combretastatin A4 inclusion complexes enable in vitro targeted cancer therapy
... The inclusion complexes of ...G5.NHAc-FI-FA/CA4 complexes was similar to that of free CA4 at the same selected drug ...the complexes were able to target selectively and display specific ...
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