[PDF] Top 20 1, 3, 4 Oxadiazole as antimicrobial agents: An overview
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1, 3, 4 Oxadiazole as antimicrobial agents: An overview
... Karthikeyan et. al.; (2008); synthesized 2,4-dichloro-5-flourophenyl containing Oxadiazoles (Compound 12 and 13) and then final compounds were tested for their antimicrobial activity. Among the tested compounds, ... See full document
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Syntheses of Substituted 1,3,4-Oxadiazole, 1,3,4-Thiadiazole and 1,2,4-Triazole Derivatives as Potential Antimicrobial Agents
... To a solution of 2 (0.01 mol) in ethanol (20 mL) alkyl (or aryl) isothiocyanate (0.01 mole) and sodium hydroxide (0.01 mol, 2 N solution) was added. The mixture was stirred for 2 h at room temperature and then acidified ... See full document
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1, 3, 4 OXADIAZOLE IN MEDICINAL CHEMISTRY: AN OVERVIEW
... ring.1,3,4 Oxadiazole are known from about eighty years and investigations in this field have intensified due to its applications in most diverse areas like dry synthesis, polymer as they give new aliphatic ... See full document
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QSRT STUDIES OF 2 (5 ARYL 1, 3, 4 OXADIAZOL 2 YL) N (5 METHYLISOXAZOL 3 YL) ACETAMIDE DERIVATIVES AS AN ANTIMICROBIAL AGENTS
... The 1, 3, 4- oxadiazoles are heterocycles of current interest due to their broad-spectrum pharmacological ...isoxazolyl 1, 3, 4-oxadiazoles have been undertaken to correlating ... See full document
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Exploration of QSAR: Oxadiazole derivatives as antimicrobial agents
... A quantitative structure activity relationship study on a series of 2, 5-(substituted) 1, 3, 4- oxadiazole analogues was made using combination of various thermodynamic, steric, electronic and ... See full document
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DOCKING STUDIES OF NOVEL 1, 3, 4- OXADIAZOLE CONTAINING 1H-INDOLE- 2, 3-DIONE ANALOGUES AS ANTICANCER PROPERTIES
... Immunotherapy has demonstrated promising results in basic and preclinical animal studies, and there have been several clinical trials in gynecologic cancer using immunologic modalities. However, clinical applications ... See full document
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SYNTHESIS & PREDICTING THE POSSIBILITY OF 2, 5 DISUBSTITUTED 1, 3, 4 OXADIAZOLE DERIVATIVES AS GSK 3β INHIBITORS
... & 4 th position of 1, 3, 4-oxadiazole when compared with the standard GSK-3beta ...disubstituted-1, 3, 4-oxadiazoles are good GSK-3beta inhibitors. These ... See full document
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Catalyst Free Synthesis of 2-(3, 4-dichlorophenyl)-1, 8a-dihydroimidazo [1, 2-a] pyridine Derivatives as Potent Antimicrobial Agents
... with antimicrobial agents, as well as patients with AIDS are immuno suppressed and very susceptible to life threatening systemic microbial infections by Candidiasis, Cryptococcoss and Aspergillosis 4,5 ... See full document
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Synthesis and Characterization of 2-phenyl-5- (1-phenyl-3-(3, 4, 5-trimethoxyphenyl)-1H-pyrazol- 4-yl) - 1, 3, 4-oxadiazole Scaffolds for Assessing Their Medicinal Potentials
... to 1 ml of poly- phenol extracts with 3 ml of ...(1, 1-dimethylethyl)-4-methylphenol (BHT) antioxidant agents was used as positive ... See full document
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DETECTION OF BACTERIAL AGENTS CAUSING URINARY TRACT INFECTION AMONG CHILDREN IN KHARTOUM STATE
... bacterial agents responsible for urinary tract infections among children from age 5-15 and the antimicrobial sensitivity profile of the uropathogens involved in these infectious ...spp 4%, ... See full document
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BENZOTRIAZOLE - OXADIAZOLE HYBRIDS AS MEDICINAL AGENTS THE SIGNIFICANCE IN UNITY IS AN ETERNAL WONDER
... novel 1, 3, 4-oxadiazole derivatives possessing benzotriazole moiety as FAK inhibitors with anticancer ...HL. 1, 3, 4-Oxadiazole derivatives as potential antitumor ... See full document
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Evaluation of Antimicrobial Profile of Some Novel 1, 3, 4-Oxadiazole Derivatives Followed by Molecular Docking Against 3G7E Bacterial DNA Gyrase
... Here we concluded that the compound AB2, AB1, AB7, AB3, AB4 and AB8 possessed potential antimicrobial activity against following bacteria: S. aureus (ATCC 9144), B. subtilis (ATCC 6633), S. epidermidis (ATCC ... See full document
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Synthesis and antimicrobial studies of 2 (5 substituted) 1, 3, 4 oxadiazole 2 yl) H imidazo [1, 2, α] pyridine derivatives
... It has long been known that imidazo [1, 2-a] pyridine derivatives exhibited diverse biological activities [1-3] and are used as antiviral, [4-12] antiulcer, [ 13-15] antibacterial, [16-17] ... See full document
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Practical use of registered veterinary medicinal products in Macedonia in identifying the risk of developing of antimicrobial resistance
... of antimicrobial agents in different therapeutic main groups (see Table 3) in order to estimate the use of antimicrobial agents in veterinary sector in the RM and to identify the risk ... See full document
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Synthesis of some novel 1, 3, 4-oxadiazole and its anti-bacterial and anti-fungal activity
... on 1, 3, 4-oxadiazole and their synthetic analogs have revealed a variety of pharmacological activities including anti-microbial, anti-tubercular and insecticidal ...activities. 1, ... See full document
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SYNTHESIS, CHARACTERIZATION AND IN VITRO ANTIINFLAMMATORY ACTIVITY OF SOME SUBSTITUTED 1, 3, 4–ARYL OXADIAZOLE DERIVATIVES
... this agents may lead to the development of gastrointestinal ulceration, bleeding and in some cases renal ...these agents had been carried ...likes antimicrobial activity [1] , ... See full document
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Synthesis and pharmacological screening of novel 6-methyl-2-oxo-4-substituted-5-(5-phenyl-1, 3, 4-oxadiazole-2yl)-1, 2, 3, 4-tetrahydropyrimidine
... Preparation of standard and test drug solutions The standard drugs and synthesized compounds were dissolved in minimum quantity of Dimethyl Formamide (DMF) and the volume is adjusted with distilled water to get 50µg/ml ... See full document
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ANTIMICROBIAL AND ANTIFUNGAL EVALUATION OF NEWLY SYNTHESIZED OXADIAZOLE DERIVATIVES BEARING 2, 4, 5 TRIPHNENYL IMIDAZOLE MOIETY
... All the chemicals used in the synthesis were supplied by E. Merck and S. D. Fine Chemicals. Melting point was determined by open capillary tube method and is uncorrected. Homogeneity of the compounds were checked on thin ... See full document
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SYNTHESIS, ANTICONVULSANT AND NEUROTOXICITY SCREENING OF SOME NOVEL 2, 5-DISUBSTITUTED - 1, 3, 4 – OXADIAZOLE DERIVATIVES
... anticonvulsant agents as it has not been possible to control every kind of seizure with currently available antiepileptic ...of oxadiazole as a basic nucleus incorporated with substituted benzoxazole moiety ... See full document
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EVALUATION OF ANTI-INFLAMMATORY AND ANALGESIC ACTIVITY OF THE NOVEL DERIVATIVES OF 1, 3, 4-OXADIAZOLE IN EXPERIMENTAL ANIMAL MODELS
... The synthesis of novel compound libraries along with screening is a rapid and effective approach for the discovery of potential chemical agents, and it becomes an important method in pharmaceutical chemistry ... See full document
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